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Assay Detail

CHEMBL1960338

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against Chinese hamster V79 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Cricetulus griseus
Cell Type V79
Confidence 1 — Organism
Curated By Autocuration

Target

V79 (CHEMBL614074)
Type CELL-LINE
Organism Cricetulus griseus

Publication

Disparate SAR data of griseofulvin analogues for the dermatophytes Trichophyton mentagrophytes, T. rubrum, and MDA-MB-231 cancer cells.
Rønnest MH, Raab MS, Anderhub S, Boesen S, Krämer A, Larsen TO, Clausen MH.
J Med Chem (2012) 55 : 652 -660
PubMed 22191585 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.63 6.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL522763 1 6.16
CHEMBL562 GRISEOFULVIN 4.0 1 5.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL522763 IC50 = 700.0 nM 6.16
CHEMBL562 GRISEOFULVIN IC50 = 8000.0 nM 5.10