Assay Detail
Binding
CHEMBL1960450
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Inhibition of rat NET-mediated uptake
2
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Wake-promoting agents: search for next generation modafinil: part II.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.73 | 4.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1956397 | — | — | 2 | 4.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1956397 | — | IC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL1956397 | — | IC50 | = | 32000.0 | nM | 4.50 |