Assay Detail
Functional
CHEMBL1963818
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: HIPK4
618
Total Activities
606
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Homeodomain-interacting protein kinase 4 (CHEMBL1075167) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 618 | 6.26 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2000335 | — | — | 1 | 8.40 |
| CHEMBL2004716 | — | — | 1 | 8.40 |
| CHEMBL411903 | — | — | 1 | 8.30 |
| CHEMBL482767 | SNS-314 | 1.0 | 1 | 8.20 |
| CHEMBL1983932 | — | — | 1 | 8.10 |
| CHEMBL1992306 | — | — | 1 | 8.00 |
| CHEMBL1988387 | — | — | 1 | 8.00 |
| CHEMBL1336 | SORAFENIB | 4.0 | 1 | 8.00 |
| CHEMBL1984162 | — | — | 1 | 8.00 |
| CHEMBL371206 | — | — | 1 | 8.00 |
| CHEMBL1982466 | — | — | 1 | 8.00 |
| CHEMBL497151 | — | — | 1 | 7.90 |
| CHEMBL2005631 | — | — | 1 | 7.90 |
| CHEMBL1979577 | — | — | 1 | 7.90 |
| CHEMBL272453 | — | — | 1 | 7.90 |
| CHEMBL1988717 | — | — | 1 | 7.90 |
| CHEMBL1967116 | — | — | 1 | 7.90 |
| CHEMBL1998585 | — | — | 1 | 7.90 |
| CHEMBL213505 | — | — | 1 | 7.90 |
| CHEMBL1970074 | — | — | 1 | 7.80 |
| CHEMBL1965988 | — | — | 1 | 7.80 |
| CHEMBL271381 | — | — | 1 | 7.80 |
| CHEMBL1973211 | — | — | 1 | 7.70 |
| CHEMBL1979883 | — | — | 1 | 7.70 |
| CHEMBL396523 | — | — | 1 | 7.70 |
| CHEMBL1980297 | ILORASERTIB | 2.0 | 1 | 7.70 |
| CHEMBL1970142 | — | — | 1 | 7.60 |
| CHEMBL1998159 | — | — | 1 | 7.60 |
| CHEMBL1989708 | — | — | 2 | 7.60 |
| CHEMBL1981725 | — | — | 1 | 7.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2000335 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL2004716 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL411903 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL482767 | SNS-314 | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1983932 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1988387 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1982466 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1336 | SORAFENIB | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1992306 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL371206 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1984162 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL2005631 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL272453 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1988717 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1998585 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1979577 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL497151 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1967116 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL213505 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1970074 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL271381 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1965988 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1980297 | ILORASERTIB | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1979883 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1973211 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL396523 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1981725 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1998159 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1989708 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1970142 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1966816 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1994321 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1973937 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL2001257 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1968406 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1979093 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1976220 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL223360 | LINIFANIB | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1982660 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1982660 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL2005828 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1989708 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1975900 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL2000801 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL1994830 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL2001751 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL196363 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL244378 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL1983025 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1980540 | — | Ki | = | 79.43 | nM | 7.10 |