Assay Detail
Functional
CHEMBL1963867
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response confirmation of uHTS hits for small molecule modulators of myocardial damage in HL-1 cells using Peroxide. (Class of assay: confirmatory)
201
Total Activities
201
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Tissue | Myocardium |
| Cell Type | HL-1 |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 201 | 4.94 | 5.83 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1884334 | — | — | 1 | 5.83 |
| CHEMBL1880550 | — | — | 1 | 5.80 |
| CHEMBL1968095 | — | — | 1 | 5.74 |
| CHEMBL1601300 | — | — | 1 | 5.74 |
| CHEMBL1448654 | — | — | 1 | 5.49 |
| CHEMBL1966961 | — | — | 1 | 5.48 |
| CHEMBL1880968 | — | — | 1 | 5.48 |
| CHEMBL1453916 | — | — | 1 | 5.46 |
| CHEMBL1725784 | — | — | 1 | 5.46 |
| CHEMBL1605288 | — | — | 1 | 5.44 |
| CHEMBL1307703 | — | — | 1 | 5.40 |
| CHEMBL1905593 | — | — | 1 | 5.39 |
| CHEMBL1431520 | — | — | 1 | 5.38 |
| CHEMBL1486891 | — | — | 1 | 5.38 |
| CHEMBL1503376 | — | — | 1 | 5.37 |
| CHEMBL1458710 | — | — | 1 | 5.37 |
| CHEMBL1343685 | — | — | 1 | 5.36 |
| CHEMBL1901953 | — | — | 1 | 5.34 |
| CHEMBL1525055 | — | — | 1 | 5.34 |
| CHEMBL1450049 | — | — | 1 | 5.27 |
| CHEMBL1718652 | — | — | 1 | 5.26 |
| CHEMBL1993796 | — | — | 1 | 5.22 |
| CHEMBL1902783 | — | — | 1 | 5.21 |
| CHEMBL1893210 | — | — | 1 | 5.21 |
| CHEMBL1894456 | — | — | 1 | 5.17 |
| CHEMBL1494757 | — | — | 1 | 5.15 |
| CHEMBL1422847 | — | — | 1 | 5.12 |
| CHEMBL1550224 | — | — | 1 | 5.07 |
| CHEMBL1547685 | — | — | 1 | 5.06 |
| CHEMBL1550633 | — | — | 1 | 5.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1884334 | — | IC50 | = | 1480.0 | nM | 5.83 |
| CHEMBL1880550 | — | IC50 | = | 1590.0 | nM | 5.80 |
| CHEMBL1968095 | — | IC50 | = | 1820.0 | nM | 5.74 |
| CHEMBL1601300 | — | IC50 | = | 1840.0 | nM | 5.74 |
| CHEMBL1448654 | — | IC50 | = | 3220.0 | nM | 5.49 |
| CHEMBL1880968 | — | IC50 | = | 3280.0 | nM | 5.48 |
| CHEMBL1966961 | — | IC50 | = | 3330.0 | nM | 5.48 |
| CHEMBL1725784 | — | IC50 | = | 3450.0 | nM | 5.46 |
| CHEMBL1453916 | — | IC50 | = | 3490.0 | nM | 5.46 |
| CHEMBL1605288 | — | IC50 | = | 3600.0 | nM | 5.44 |
| CHEMBL1307703 | — | IC50 | = | 3990.0 | nM | 5.40 |
| CHEMBL1905593 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL1431520 | — | IC50 | = | 4130.0 | nM | 5.38 |
| CHEMBL1486891 | — | IC50 | = | 4220.0 | nM | 5.38 |
| CHEMBL1458710 | — | IC50 | = | 4320.0 | nM | 5.37 |
| CHEMBL1503376 | — | IC50 | = | 4240.0 | nM | 5.37 |
| CHEMBL1343685 | — | IC50 | = | 4350.0 | nM | 5.36 |
| CHEMBL1901953 | — | IC50 | = | 4550.0 | nM | 5.34 |
| CHEMBL1525055 | — | IC50 | = | 4530.0 | nM | 5.34 |
| CHEMBL1450049 | — | IC50 | = | 5410.0 | nM | 5.27 |
| CHEMBL1718652 | — | IC50 | = | 5510.0 | nM | 5.26 |
| CHEMBL1993796 | — | IC50 | = | 6020.0 | nM | 5.22 |
| CHEMBL1902783 | — | IC50 | = | 6110.0 | nM | 5.21 |
| CHEMBL1893210 | — | IC50 | = | 6150.0 | nM | 5.21 |
| CHEMBL1894456 | — | IC50 | = | 6830.0 | nM | 5.17 |
| CHEMBL1494757 | — | IC50 | = | 7020.0 | nM | 5.15 |
| CHEMBL1422847 | — | IC50 | = | 7510.0 | nM | 5.12 |
| CHEMBL1550224 | — | IC50 | = | 8500.0 | nM | 5.07 |
| CHEMBL1879313 | — | IC50 | = | 8730.0 | nM | 5.06 |
| CHEMBL1547685 | — | IC50 | = | 8710.0 | nM | 5.06 |
| CHEMBL1550633 | — | IC50 | = | 8630.0 | nM | 5.06 |
| CHEMBL1967640 | — | IC50 | = | 9150.0 | nM | 5.04 |
| CHEMBL1385111 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL1421091 | — | IC50 | = | 10400.0 | nM | 4.98 |
| CHEMBL1969457 | — | IC50 | = | 10900.0 | nM | 4.96 |
| CHEMBL1878680 | — | IC50 | = | 11600.0 | nM | 4.94 |
| CHEMBL1904672 | — | IC50 | = | 11430.0 | nM | 4.94 |
| CHEMBL1722488 | — | IC50 | = | 11700.0 | nM | 4.93 |
| CHEMBL1319264 | — | IC50 | = | 11930.0 | nM | 4.92 |
| CHEMBL1545153 | — | IC50 | = | 12140.0 | nM | 4.92 |
| CHEMBL1880473 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL1364287 | — | IC50 | = | 12350.0 | nM | 4.91 |
| CHEMBL1713021 | — | IC50 | = | 12700.0 | nM | 4.90 |
| CHEMBL1867718 | — | IC50 | = | 12900.0 | nM | 4.89 |
| CHEMBL1459314 | — | IC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL1602676 | — | IC50 | = | 13800.0 | nM | 4.86 |
| CHEMBL1559375 | — | IC50 | = | 13700.0 | nM | 4.86 |
| CHEMBL1475866 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL1888730 | — | IC50 | = | 15050.0 | nM | 4.82 |
| CHEMBL1505748 | — | IC50 | = | 15900.0 | nM | 4.80 |