Assay Detail
Functional
CHEMBL1963907
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: TRFRET-based biochemical high throughput dose response assay for inhibitors of the interaction of the Ras and Rab interactor 1 protein (Rin1) and the c-abl oncogene 1, non-receptor tyrosine kinase (Abl). (Class of assay: confirmatory)
230
Total Activities
229
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Target
Ras and Rab interactor 1/Tyrosine-protein kinase ABL1 (CHEMBL3885630) ↗| Type | PROTEIN-PROTEIN INTERACTION |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 230 | 5.16 | 8.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1608529 | — | — | 1 | 8.05 |
| CHEMBL1232381 | — | — | 1 | 8.00 |
| CHEMBL1504308 | — | — | 1 | 7.85 |
| CHEMBL1343539 | — | — | 1 | 7.84 |
| CHEMBL1399113 | — | — | 1 | 7.82 |
| CHEMBL1403262 | — | — | 1 | 7.76 |
| CHEMBL1311154 | — | — | 1 | 7.73 |
| CHEMBL1475400 | — | — | 1 | 7.58 |
| CHEMBL1417216 | — | — | 1 | 7.01 |
| CHEMBL1369512 | — | — | 1 | 6.97 |
| CHEMBL1455014 | — | — | 1 | 6.72 |
| CHEMBL601757 | — | — | 1 | 6.52 |
| CHEMBL578512 | — | — | 1 | 6.49 |
| CHEMBL1356021 | — | — | 1 | 6.39 |
| CHEMBL1732813 | — | — | 1 | 6.29 |
| CHEMBL1325945 | — | — | 1 | 6.28 |
| CHEMBL857 | BIOTIN | 4.0 | 2 | 6.28 |
| CHEMBL1369913 | — | — | 1 | 6.26 |
| CHEMBL1512846 | — | — | 1 | 6.21 |
| CHEMBL1580441 | — | — | 1 | 6.18 |
| CHEMBL1501047 | — | — | 1 | 6.16 |
| CHEMBL1571034 | — | — | 1 | 6.14 |
| CHEMBL175266 | — | — | 1 | 6.08 |
| CHEMBL1336319 | — | — | 1 | 6.04 |
| CHEMBL1485830 | — | — | 1 | 5.99 |
| CHEMBL1896885 | — | — | 1 | 5.90 |
| CHEMBL1722228 | — | — | 1 | 5.87 |
| CHEMBL1736479 | — | — | 1 | 5.86 |
| CHEMBL1303555 | — | — | 1 | 5.85 |
| CHEMBL1565528 | — | — | 1 | 5.84 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1608529 | — | IC50 | = | 8.97 | nM | 8.05 |
| CHEMBL1232381 | — | IC50 | = | 10.06 | nM | 8.00 |
| CHEMBL1504308 | — | IC50 | = | 14.27 | nM | 7.85 |
| CHEMBL1343539 | — | IC50 | = | 14.53 | nM | 7.84 |
| CHEMBL1399113 | — | IC50 | = | 15.03 | nM | 7.82 |
| CHEMBL1403262 | — | IC50 | = | 17.35 | nM | 7.76 |
| CHEMBL1311154 | — | IC50 | = | 18.69 | nM | 7.73 |
| CHEMBL1475400 | — | IC50 | = | 26.15 | nM | 7.58 |
| CHEMBL1417216 | — | IC50 | = | 96.68 | nM | 7.01 |
| CHEMBL1369512 | — | IC50 | = | 106.16 | nM | 6.97 |
| CHEMBL1455014 | — | IC50 | = | 191.92 | nM | 6.72 |
| CHEMBL601757 | — | IC50 | = | 302.03 | nM | 6.52 |
| CHEMBL578512 | — | IC50 | = | 323.05 | nM | 6.49 |
| CHEMBL1356021 | — | IC50 | = | 406.94 | nM | 6.39 |
| CHEMBL1732813 | — | IC50 | = | 514.16 | nM | 6.29 |
| CHEMBL1325945 | — | IC50 | = | 527.38 | nM | 6.28 |
| CHEMBL857 | BIOTIN | IC50 | = | 528.66 | nM | 6.28 |
| CHEMBL1369913 | — | IC50 | = | 548.02 | nM | 6.26 |
| CHEMBL1512846 | — | IC50 | = | 618.21 | nM | 6.21 |
| CHEMBL1580441 | — | IC50 | = | 659.08 | nM | 6.18 |
| CHEMBL1501047 | — | IC50 | = | 695.03 | nM | 6.16 |
| CHEMBL1571034 | — | IC50 | = | 724.16 | nM | 6.14 |
| CHEMBL175266 | — | IC50 | = | 834.68 | nM | 6.08 |
| CHEMBL1336319 | — | IC50 | = | 905.0 | nM | 6.04 |
| CHEMBL1485830 | — | IC50 | = | 1025.0 | nM | 5.99 |
| CHEMBL1896885 | — | IC50 | = | 1268.0 | nM | 5.90 |
| CHEMBL1722228 | — | IC50 | = | 1346.0 | nM | 5.87 |
| CHEMBL1736479 | — | IC50 | = | 1378.0 | nM | 5.86 |
| CHEMBL1303555 | — | IC50 | = | 1405.0 | nM | 5.85 |
| CHEMBL1565528 | — | IC50 | = | 1451.0 | nM | 5.84 |
| CHEMBL1892599 | — | IC50 | = | 1536.0 | nM | 5.81 |
| CHEMBL1441033 | — | IC50 | = | 1679.0 | nM | 5.78 |
| CHEMBL1607186 | — | IC50 | = | 1857.0 | nM | 5.73 |
| CHEMBL1704366 | — | IC50 | = | 1863.0 | nM | 5.73 |
| CHEMBL1335745 | — | IC50 | = | 1899.0 | nM | 5.72 |
| CHEMBL1868487 | — | IC50 | = | 1896.0 | nM | 5.72 |
| CHEMBL1554805 | — | IC50 | = | 2032.0 | nM | 5.69 |
| CHEMBL1348125 | — | IC50 | = | 2187.0 | nM | 5.66 |
| CHEMBL1718137 | — | IC50 | = | 2218.0 | nM | 5.65 |
| CHEMBL156383 | — | IC50 | = | 2330.0 | nM | 5.63 |
| CHEMBL1585699 | — | IC50 | = | 2386.0 | nM | 5.62 |
| CHEMBL1551052 | — | IC50 | = | 2484.0 | nM | 5.61 |
| CHEMBL1407551 | — | IC50 | = | 2621.0 | nM | 5.58 |
| CHEMBL1560085 | — | IC50 | = | 2867.0 | nM | 5.54 |
| CHEMBL1972558 | — | IC50 | = | 2939.0 | nM | 5.53 |
| CHEMBL1611726 | — | IC50 | = | 2997.0 | nM | 5.52 |
| CHEMBL1863690 | — | IC50 | = | 3139.0 | nM | 5.50 |
| CHEMBL1350329 | — | IC50 | = | 3229.0 | nM | 5.49 |
| CHEMBL1329549 | — | IC50 | = | 3458.0 | nM | 5.46 |
| CHEMBL2000834 | — | IC50 | = | 3590.0 | nM | 5.45 |