Assay Detail
Binding
CHEMBL2015428
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Binding affinity to C-terminus C9-tagged immobilized CCR5 by SPR analysis
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Screening for GPCR Ligands Using Surface Plasmon Resonance.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 7 | 4.73 | 5.09 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2011439 | — | — | 1 | 5.09 |
| CHEMBL1618631 | — | — | 1 | 5.00 |
| CHEMBL2011440 | — | — | 1 | 4.76 |
| CHEMBL1907216 | — | — | 1 | 4.74 |
| CHEMBL2011441 | — | — | 1 | 4.65 |
| CHEMBL1623307 | — | — | 1 | 4.56 |
| CHEMBL1621896 | — | — | 1 | 4.31 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2011439 | — | Kd | = | 8200.0 | nM | 5.09 |
| CHEMBL1618631 | — | Kd | = | 10000.0 | nM | 5.00 |
| CHEMBL2011440 | — | Kd | = | 17500.0 | nM | 4.76 |
| CHEMBL1907216 | — | Kd | = | 18400.0 | nM | 4.74 |
| CHEMBL2011441 | — | Kd | = | 22600.0 | nM | 4.65 |
| CHEMBL1623307 | — | Kd | = | 27500.0 | nM | 4.56 |
| CHEMBL1621896 | — | Kd | = | 49000.0 | nM | 4.31 |