Assay Detail
Binding
CHEMBL2033711
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Inhibition of human ABL by radiometric assay
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Multiple determinants for selective inhibition of apicomplexan calcium-dependent protein kinase CDPK1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 16 | 5.88 | 7.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1241489 | — | — | 1 | 7.16 |
| CHEMBL2030556 | — | — | 1 | 6.55 |
| CHEMBL1785020 | — | — | 1 | 6.12 |
| CHEMBL1785021 | — | — | 1 | 5.80 |
| CHEMBL1242754 | — | — | 1 | 5.80 |
| CHEMBL685 | MEBENDAZOLE | 4.0 | 1 | 5.34 |
| CHEMBL2030558 | — | — | 1 | 5.26 |
| CHEMBL2030560 | — | — | 1 | 5.00 |
| CHEMBL2030552 | — | — | 1 | - |
| CHEMBL2030553 | — | — | 1 | - |
| CHEMBL2030554 | — | — | 1 | - |
| CHEMBL2030555 | — | — | 1 | - |
| CHEMBL2030557 | — | — | 1 | - |
| CHEMBL1785018 | — | — | 1 | - |
| CHEMBL2030559 | — | — | 1 | - |
| CHEMBL2030561 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1241489 | — | Ki | = | 69.0 | nM | 7.16 |
| CHEMBL2030556 | — | Ki | = | 280.0 | nM | 6.55 |
| CHEMBL1785020 | — | Ki | = | 750.0 | nM | 6.12 |
| CHEMBL1785021 | — | Ki | = | 1600.0 | nM | 5.80 |
| CHEMBL1242754 | — | Ki | = | 1600.0 | nM | 5.80 |
| CHEMBL685 | MEBENDAZOLE | Ki | = | 4600.0 | nM | 5.34 |
| CHEMBL2030558 | — | Ki | = | 5500.0 | nM | 5.26 |
| CHEMBL2030560 | — | Ki | = | 10000.0 | nM | 5.00 |
| CHEMBL2030552 | — | Ki | - | — | - | |
| CHEMBL2030553 | — | Ki | > | 15000.0 | nM | - |
| CHEMBL2030554 | — | Ki | > | 15000.0 | nM | - |
| CHEMBL2030555 | — | Ki | > | 15000.0 | nM | - |
| CHEMBL2030557 | — | Ki | - | — | - | |
| CHEMBL1785018 | — | Ki | - | — | - | |
| CHEMBL2030559 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL2030561 | — | Ki | > | 10000.0 | nM | - |