Assay Detail
Binding
CHEMBL2034616
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to rabbit muscular GPa by NMR binding assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Oryctolagus cuniculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Glycogen phosphorylase, muscle form (CHEMBL4696) ↗| Type | SINGLE PROTEIN |
| Organism | Oryctolagus cuniculus |
Publication
Binding evaluation of fragment-based scaffolds for probing allosteric enzymes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 4.98 | 5.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2030483 | — | — | 1 | 5.57 |
| CHEMBL337309 | TAXIFOLIN | — | 1 | 5.32 |
| CHEMBL2030484 | — | — | 1 | 5.00 |
| CHEMBL277157 | — | — | 1 | 4.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2030483 | — | IC50 | = | 2700.0 | nM | 5.57 |
| CHEMBL337309 | TAXIFOLIN | IC50 | = | 4800.0 | nM | 5.32 |
| CHEMBL2030484 | — | IC50 | = | 9900.0 | nM | 5.00 |
| CHEMBL277157 | — | IC50 | = | 96900.0 | nM | 4.01 |