Assay Detail
Functional
CHEMBL2038470
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiobesity activity in po dosed fasted rat assessed as reduction in TAG to DAG ratio in adipose tissue
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Tissue | Adipose tissue |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Identification, optimisation and in vivo evaluation of oxadiazole DGAT-1 inhibitors for the treatment of obesity and diabetes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 9.52 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2036730 | — | — | 1 | 9.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2036730 | — | IC50 | = | 0.3 | nM | 9.52 |