Assay Detail
Functional
CHEMBL2040652
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Plaque growth inhibition
48
Total Activities
48
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Canis lupus familiaris |
| Cell Type | MDCK |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Polymerase acidic protein (CHEMBL1169598) ↗| Type | SINGLE PROTEIN |
| Organism | Influenza A virus (A/Puerto Rico/8/1934(H1N1)) |
Publication
Identification of influenza endonuclease inhibitors using a novel fluorescence polarization assay.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 48 | 5.15 | 6.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2040554 | — | — | 1 | 6.10 |
| CHEMBL463590 | — | — | 1 | 6.07 |
| CHEMBL573638 | — | — | 1 | 5.84 |
| CHEMBL2040552 | — | — | 1 | 5.82 |
| CHEMBL2040581 | — | — | 1 | 5.82 |
| CHEMBL467389 | — | — | 1 | 5.68 |
| CHEMBL16755 | — | — | 1 | 5.49 |
| CHEMBL2040578 | — | — | 1 | 5.46 |
| CHEMBL2040584 | — | — | 1 | 5.46 |
| CHEMBL1829211 | — | — | 1 | 5.45 |
| CHEMBL2040569 | — | — | 1 | 5.44 |
| CHEMBL2040576 | — | — | 1 | 5.43 |
| CHEMBL205130 | — | — | 1 | 5.42 |
| CHEMBL2040583 | — | — | 1 | 5.31 |
| CHEMBL2040574 | — | — | 1 | 5.27 |
| CHEMBL2040582 | — | — | 1 | 5.26 |
| CHEMBL181602 | — | — | 1 | 5.23 |
| CHEMBL1829214 | — | — | 1 | 5.17 |
| CHEMBL492768 | — | — | 1 | 5.17 |
| CHEMBL2040553 | — | — | 1 | 5.17 |
| CHEMBL2040580 | — | — | 1 | 5.12 |
| CHEMBL2040555 | — | — | 1 | 5.09 |
| CHEMBL2040573 | — | — | 1 | 4.94 |
| CHEMBL2040563 | — | — | 1 | 4.74 |
| CHEMBL2040575 | — | — | 1 | 4.65 |
| CHEMBL2040585 | — | — | 1 | 4.61 |
| CHEMBL2040568 | — | — | 1 | 4.59 |
| CHEMBL2040577 | — | — | 1 | 4.45 |
| CHEMBL2040562 | — | — | 1 | 4.23 |
| CHEMBL2040561 | — | — | 1 | 4.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2040554 | — | EC50 | = | 800.0 | nM | 6.10 |
| CHEMBL463590 | — | EC50 | = | 860.0 | nM | 6.07 |
| CHEMBL573638 | — | EC50 | = | 1450.0 | nM | 5.84 |
| CHEMBL2040552 | — | EC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL2040581 | — | EC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL467389 | — | EC50 | = | 2070.0 | nM | 5.68 |
| CHEMBL16755 | — | EC50 | = | 3220.0 | nM | 5.49 |
| CHEMBL2040578 | — | EC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL2040584 | — | EC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL1829211 | — | EC50 | = | 3560.0 | nM | 5.45 |
| CHEMBL2040569 | — | EC50 | = | 3660.0 | nM | 5.44 |
| CHEMBL2040576 | — | EC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL205130 | — | EC50 | = | 3800.0 | nM | 5.42 |
| CHEMBL2040583 | — | EC50 | = | 4851.0 | nM | 5.31 |
| CHEMBL2040574 | — | EC50 | = | 5410.0 | nM | 5.27 |
| CHEMBL2040582 | — | EC50 | = | 5520.0 | nM | 5.26 |
| CHEMBL181602 | — | EC50 | = | 5920.0 | nM | 5.23 |
| CHEMBL1829214 | — | EC50 | = | 6800.0 | nM | 5.17 |
| CHEMBL492768 | — | EC50 | = | 6800.0 | nM | 5.17 |
| CHEMBL2040553 | — | EC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL2040580 | — | EC50 | = | 7670.0 | nM | 5.12 |
| CHEMBL2040555 | — | EC50 | = | 8170.0 | nM | 5.09 |
| CHEMBL2040573 | — | EC50 | = | 11480.0 | nM | 4.94 |
| CHEMBL2040563 | — | EC50 | = | 18090.0 | nM | 4.74 |
| CHEMBL2040575 | — | EC50 | = | 22600.0 | nM | 4.65 |
| CHEMBL2040585 | — | EC50 | = | 24300.0 | nM | 4.61 |
| CHEMBL2040568 | — | EC50 | = | 25460.0 | nM | 4.59 |
| CHEMBL2040577 | — | EC50 | = | 35300.0 | nM | 4.45 |
| CHEMBL2040562 | — | EC50 | = | 58900.0 | nM | 4.23 |
| CHEMBL2040561 | — | EC50 | = | 67400.0 | nM | 4.17 |
| CHEMBL2040564 | — | EC50 | = | 71300.0 | nM | 4.15 |
| CHEMBL2040570 | — | EC50 | = | 88120.0 | nM | 4.05 |
| CHEMBL2040566 | — | EC50 | = | 151800.0 | nM | - |
| CHEMBL2040567 | — | EC50 | = | 119700.0 | nM | - |
| CHEMBL2040571 | — | EC50 | = | 216700.0 | nM | - |
| CHEMBL2040572 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL424 | SALICYLIC ACID | EC50 | > | 250000.0 | nM | - |
| CHEMBL2040565 | — | EC50 | = | 156100.0 | nM | - |
| CHEMBL2040560 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL461681 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL2040579 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL16365 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL2040559 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL456227 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL2040558 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL2040557 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL2040556 | — | EC50 | > | 250000.0 | nM | - |
| CHEMBL374569 | — | EC50 | > | 250000.0 | nM | - |