Assay Detail
Binding
CHEMBL2065345
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Inhibition of CDC7
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Cell division cycle 7-related protein kinase (CHEMBL5443) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Targeted kinase selectivity from kinase profiling data.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 9.43 | 9.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2062936 | — | — | 1 | 9.80 |
| CHEMBL2062937 | — | — | 1 | 9.50 |
| CHEMBL1999931 | — | — | 1 | 9.30 |
| CHEMBL1983595 | — | — | 1 | 9.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2062936 | — | Ki | = | 0.1585 | nM | 9.80 |
| CHEMBL2062937 | — | Ki | = | 0.3162 | nM | 9.50 |
| CHEMBL1999931 | — | Ki | = | 0.5012 | nM | 9.30 |
| CHEMBL1983595 | — | Ki | = | 0.7943 | nM | 9.10 |