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Assay Detail

CHEMBL2072274

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of 3[H]R-PIA from human A1 adenosine receptor expressed in CHO cells after 60 mins by Liquid scintillation analysis
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Adenosine receptor A1 (CHEMBL226)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Optimization of adenosine 5'-carboxamide derivatives as adenosine receptor agonists using structure-based ligand design and fragment screening.
Tosh DK, Phan K, Gao ZG, Gakh AA, Xu F, Deflorian F, Abagyan R, Stevens RC, Jacobson KA, Katritch V.
J Med Chem (2012) 55 : 4297 -4308
PubMed 22486652 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 8 8.10 8.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL261482 1 8.72
CHEMBL464859 NECA 1 8.52
CHEMBL2070507 1 8.26
CHEMBL1235128 1 7.92
CHEMBL1234591 1 7.89
CHEMBL2070398 1 7.82
CHEMBL2070508 1 7.57
CHEMBL2070506 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL261482 Ki = 1.9 nM 8.72
CHEMBL464859 NECA Ki = 3.0 nM 8.52
CHEMBL2070507 Ki = 5.5 nM 8.26
CHEMBL1235128 Ki = 12.0 nM 7.92
CHEMBL1234591 Ki = 12.8 nM 7.89
CHEMBL2070398 Ki = 15.0 nM 7.82
CHEMBL2070508 Ki = 27.0 nM 7.57
CHEMBL2070506 Ki > 10000.0 nM -