Assay Detail
Functional
CHEMBL2154227
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Cytotoxicity against human MDA-MB-361 cells after 3 days by SRB assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MDA-MB-361 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis, anticancer activities and molecular modeling studies of novel indole retinoid derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.00 | 7.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2153844 | — | — | 1 | 7.22 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 6.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2153844 | — | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 170.0 | nM | 6.77 |