Assay Detail
Binding
CHEMBL2155055
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]-DAMGO from mouse MOR/DOR expressed in HEK293 cells
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | HEK293 |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Tuned-Affinity Bivalent Ligands for the Characterization of Opioid Receptor Heteromers.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 9 | 7.78 | 9.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL19019 | NALTREXONE | 4.0 | 1 | 9.06 |
| CHEMBL1237164 | NALTRINDOLE HYDROCHLORIDE | — | 1 | 8.46 |
| CHEMBL2151247 | — | — | 1 | 8.38 |
| CHEMBL963 | OXYMORPHONE | 4.0 | 1 | 8.33 |
| CHEMBL2151327 | — | — | 1 | 8.21 |
| CHEMBL2151328 | — | — | 1 | 6.94 |
| CHEMBL2151248 | — | — | 1 | 6.90 |
| CHEMBL2151246 | — | — | 1 | 5.92 |
| CHEMBL2151245 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL19019 | NALTREXONE | Ki | = | 0.871 | nM | 9.06 |
| CHEMBL1237164 | NALTRINDOLE HYDROCHLORIDE | Ki | = | 3.467 | nM | 8.46 |
| CHEMBL2151247 | — | Ki | = | 4.169 | nM | 8.38 |
| CHEMBL963 | OXYMORPHONE | Ki | = | 4.677 | nM | 8.33 |
| CHEMBL2151327 | — | Ki | = | 6.166 | nM | 8.21 |
| CHEMBL2151328 | — | Ki | = | 114.82 | nM | 6.94 |
| CHEMBL2151248 | — | Ki | = | 125.89 | nM | 6.90 |
| CHEMBL2151246 | — | Ki | = | 1202.26 | nM | 5.92 |
| CHEMBL2151245 | — | Ki | < | 1.0 | nM | - |