Assay Detail
Functional
CHEMBL2155897
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Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysis
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 15 | 9.80 | 10.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2151643 | — | — | 1 | 10.39 |
| CHEMBL376756 | KISSPEPTIN-10 | 3.0 | 1 | 10.31 |
| CHEMBL2151646 | — | — | 1 | 10.30 |
| CHEMBL2151642 | — | — | 1 | 10.19 |
| CHEMBL2151654 | — | — | 1 | 10.14 |
| CHEMBL2151653 | — | — | 1 | 10.01 |
| CHEMBL2151650 | — | — | 1 | 10.00 |
| CHEMBL2151652 | — | — | 1 | 9.96 |
| CHEMBL2151649 | — | — | 1 | 9.89 |
| CHEMBL2151648 | — | — | 1 | 9.62 |
| CHEMBL2151651 | — | — | 1 | 9.62 |
| CHEMBL2151655 | — | — | 1 | 9.23 |
| CHEMBL2151644 | — | — | 1 | 9.21 |
| CHEMBL2151647 | — | — | 1 | 9.14 |
| CHEMBL2151645 | — | — | 1 | 9.02 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2151643 | — | EC50 | = | 0.041 | nM | 10.39 |
| CHEMBL376756 | KISSPEPTIN-10 | EC50 | = | 0.049 | nM | 10.31 |
| CHEMBL2151646 | — | EC50 | = | 0.05 | nM | 10.30 |
| CHEMBL2151642 | — | EC50 | = | 0.065 | nM | 10.19 |
| CHEMBL2151654 | — | EC50 | = | 0.072 | nM | 10.14 |
| CHEMBL2151653 | — | EC50 | = | 0.098 | nM | 10.01 |
| CHEMBL2151650 | — | EC50 | = | 0.1 | nM | 10.00 |
| CHEMBL2151652 | — | EC50 | = | 0.11 | nM | 9.96 |
| CHEMBL2151649 | — | EC50 | = | 0.13 | nM | 9.89 |
| CHEMBL2151648 | — | EC50 | = | 0.24 | nM | 9.62 |
| CHEMBL2151651 | — | EC50 | = | 0.24 | nM | 9.62 |
| CHEMBL2151655 | — | EC50 | = | 0.59 | nM | 9.23 |
| CHEMBL2151644 | — | EC50 | = | 0.62 | nM | 9.21 |
| CHEMBL2151647 | — | EC50 | = | 0.73 | nM | 9.14 |
| CHEMBL2151645 | — | EC50 | = | 0.95 | nM | 9.02 |