Assay Detail
Binding
CHEMBL2168070
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human recombinant FAAH
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of potent inhibitors of human and mouse fatty acid amide hydrolases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 23 | 6.85 | 7.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL451909 | — | — | 1 | 7.44 |
| CHEMBL2165094 | — | — | 1 | 6.99 |
| CHEMBL2165083 | — | — | 1 | 6.77 |
| CHEMBL177577 | — | — | 1 | 6.20 |
| CHEMBL2165075 | — | — | 1 | - |
| CHEMBL2165074 | — | — | 1 | - |
| CHEMBL2165073 | — | — | 1 | - |
| CHEMBL2165072 | — | — | 1 | - |
| CHEMBL2165071 | — | — | 1 | - |
| CHEMBL2165070 | — | — | 1 | - |
| CHEMBL2165093 | — | — | 1 | - |
| CHEMBL2165092 | — | — | 1 | - |
| CHEMBL2165091 | — | — | 1 | - |
| CHEMBL2165076 | — | — | 1 | - |
| CHEMBL2165089 | — | — | 1 | - |
| CHEMBL2165088 | — | — | 1 | - |
| CHEMBL2165087 | — | — | 1 | - |
| CHEMBL2165086 | — | — | 1 | - |
| CHEMBL2165085 | — | — | 1 | - |
| CHEMBL2165084 | — | — | 1 | - |
| CHEMBL2165082 | — | — | 1 | - |
| CHEMBL2165095 | — | — | 1 | - |
| CHEMBL2165090 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL451909 | — | IC50 | = | 36.0 | nM | 7.44 |
| CHEMBL2165094 | — | IC50 | = | 102.0 | nM | 6.99 |
| CHEMBL2165083 | — | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL177577 | — | IC50 | = | 628.0 | nM | 6.20 |
| CHEMBL2165075 | — | IC50 | - | — | - | |
| CHEMBL2165074 | — | IC50 | - | — | - | |
| CHEMBL2165073 | — | IC50 | - | — | - | |
| CHEMBL2165072 | — | IC50 | - | — | - | |
| CHEMBL2165071 | — | IC50 | - | — | - | |
| CHEMBL2165070 | — | IC50 | - | — | - | |
| CHEMBL2165093 | — | IC50 | - | — | - | |
| CHEMBL2165092 | — | IC50 | - | — | - | |
| CHEMBL2165091 | — | IC50 | - | — | - | |
| CHEMBL2165076 | — | IC50 | - | — | - | |
| CHEMBL2165089 | — | IC50 | - | — | - | |
| CHEMBL2165088 | — | IC50 | - | — | - | |
| CHEMBL2165087 | — | IC50 | - | — | - | |
| CHEMBL2165086 | — | IC50 | - | — | - | |
| CHEMBL2165085 | — | IC50 | - | — | - | |
| CHEMBL2165084 | — | IC50 | - | — | - | |
| CHEMBL2165082 | — | IC50 | - | — | - | |
| CHEMBL2165095 | — | IC50 | - | — | - | |
| CHEMBL2165090 | — | IC50 | - | — | - |