Assay Detail
Binding
CHEMBL2168890
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]2-chloro-N6-cyclopentyladenosine from human A2AR
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Orally active adenosine A(1) receptor agonists with antinociceptive effects in mice.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.57 | 5.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2163560 | — | — | 1 | 5.80 |
| CHEMBL2163561 | — | — | 1 | 5.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2163560 | — | Ki | = | 1600.0 | nM | 5.80 |
| CHEMBL2163561 | — | Ki | = | 4700.0 | nM | 5.33 |