Assay Detail
Binding
CHEMBL2173154
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of CDPK4 in Plasmodium falciparum 3D7 microgametes
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Plasmodium falciparum |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Calcium-dependent protein kinase 4 (CHEMBL2169725) ↗| Type | SINGLE PROTEIN |
| Organism | Plasmodium falciparum (isolate 3D7) |
Publication
Recent results in protein kinase inhibition for tropical diseases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.58 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2030554 | — | — | 1 | 8.40 |
| CHEMBL1231371 | — | — | 1 | 6.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2030554 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL1231371 | — | IC50 | = | 177.0 | nM | 6.75 |