Assay Detail
Binding
CHEMBL2173907
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Binding affinity to human recombinant 5HT1A receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Mitigating heterocycle metabolism in drug discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.99 | 9.07 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL300739 | — | — | 1 | 9.07 |
| CHEMBL300100 | — | — | 1 | 8.90 |
| CHEMBL51457 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL300739 | — | Ki | = | 0.8511 | nM | 9.07 |
| CHEMBL300100 | — | Ki | = | 1.259 | nM | 8.90 |
| CHEMBL51457 | — | Ki | = | 436515832.24 | nM | - |