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Assay Detail

CHEMBL2174885

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cells after 60 min Packard Cobra 2 gamma-counter
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Adenosine receptor A3 (CHEMBL256)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Structural sweet spot for A1 adenosine receptor activation by truncated (N)-methanocarba nucleosides: receptor docking and potent anticonvulsant activity.
Tosh DK, Paoletta S, Deflorian F, Phan K, Moss SM, Gao ZG, Jiang X, Jacobson KA.
J Med Chem (2012) 55 : 8075 -8090
PubMed 22921089 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 22 6.47 8.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2012684 1 8.05
CHEMBL1512545 1 7.91
CHEMBL2170795 1 7.77
CHEMBL2170797 1 7.16
CHEMBL2012685 1 6.96
CHEMBL2170785 1 6.82
CHEMBL2012672 1 6.80
CHEMBL2170796 1 6.74
CHEMBL2012686 1 6.33
CHEMBL2170798 1 6.31
CHEMBL2170792 1 6.26
CHEMBL2012680 1 6.22
CHEMBL2170799 1 6.19
CHEMBL2170800 1 6.17
CHEMBL2170787 1 6.11
CHEMBL2170786 1 6.11
CHEMBL2170793 1 6.10
CHEMBL2170788 1 5.76
CHEMBL2170791 1 5.75
CHEMBL2170794 1 5.66
CHEMBL2170790 1 5.55
CHEMBL2170789 1 5.53

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2012684 Ki = 8.9 nM 8.05
CHEMBL1512545 Ki = 12.4 nM 7.91
CHEMBL2170795 Ki = 17.0 nM 7.77
CHEMBL2170797 Ki = 70.0 nM 7.16
CHEMBL2012685 Ki = 110.0 nM 6.96
CHEMBL2170785 Ki = 150.0 nM 6.82
CHEMBL2012672 Ki = 160.0 nM 6.80
CHEMBL2170796 Ki = 182.0 nM 6.74
CHEMBL2012686 Ki = 470.0 nM 6.33
CHEMBL2170798 Ki = 490.0 nM 6.31
CHEMBL2170792 Ki = 550.0 nM 6.26
CHEMBL2012680 Ki = 606.0 nM 6.22
CHEMBL2170799 Ki = 640.0 nM 6.19
CHEMBL2170800 Ki = 670.0 nM 6.17
CHEMBL2170787 Ki = 780.0 nM 6.11
CHEMBL2170786 Ki = 780.0 nM 6.11
CHEMBL2170793 Ki = 790.0 nM 6.10
CHEMBL2170788 Ki = 1720.0 nM 5.76
CHEMBL2170791 Ki = 1760.0 nM 5.75
CHEMBL2170794 Ki = 2200.0 nM 5.66
CHEMBL2170790 Ki = 2790.0 nM 5.55
CHEMBL2170789 Ki = 2930.0 nM 5.53