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Assay Detail

CHEMBL2175142

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain homogenates
24
Total Activities
24
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Cavia porcellus
Tissue Brain
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Sigma non-opioid intracellular receptor 1 (CHEMBL4153)
Type SINGLE PROTEIN
Organism Cavia porcellus

Publication

Enantiomerically pure 1,3-dioxanes as highly selective NMDA and σ₁ receptor ligands.
Köhler J, Bergander K, Fabian J, Schepmann D, Wünsch B.
J Med Chem (2012) 55 : 8953 -8957
PubMed 23013229 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 24 7.54 8.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1783450 1 8.22
CHEMBL54 HALOPERIDOL 4.0 1 8.22
CHEMBL60542 (+)-PENTAZOCINE 1 8.22
CHEMBL2170313 1 7.96
CHEMBL2170314 1 7.77
CHEMBL1783458 1 7.70
CHEMBL2170178 1 7.55
CHEMBL2170312 1 7.30
CHEMBL2170180 1 7.14
CHEMBL2170302 1 6.89
CHEMBL2170179 1 6.87
CHEMBL2170301 1 6.60
CHEMBL2170303 1 -
CHEMBL2170311 1 -
CHEMBL2170310 1 -
CHEMBL2170309 1 -
CHEMBL2170308 1 -
CHEMBL1783455 1 -
CHEMBL2170307 1 -
CHEMBL2170306 1 -
CHEMBL2170305 1 -
CHEMBL1783426 1 -
CHEMBL2170304 1 -
CHEMBL2170315 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1783450 Ki = 6.0 nM 8.22
CHEMBL54 HALOPERIDOL Ki = 6.0 nM 8.22
CHEMBL60542 (+)-PENTAZOCINE Ki = 6.0 nM 8.22
CHEMBL2170313 Ki = 11.0 nM 7.96
CHEMBL2170314 Ki = 17.0 nM 7.77
CHEMBL1783458 Ki = 20.0 nM 7.70
CHEMBL2170178 Ki = 28.0 nM 7.55
CHEMBL2170312 Ki = 50.0 nM 7.30
CHEMBL2170180 Ki = 72.0 nM 7.14
CHEMBL2170302 Ki = 128.0 nM 6.89
CHEMBL2170179 Ki = 136.0 nM 6.87
CHEMBL2170301 Ki = 253.0 nM 6.60
CHEMBL2170303 Ki > 10000.0 nM -
CHEMBL2170311 Ki > 10000.0 nM -
CHEMBL2170310 Ki > 10000.0 nM -
CHEMBL2170309 Ki > 10000.0 nM -
CHEMBL2170308 Ki > 10000.0 nM -
CHEMBL1783455 Ki > 10000.0 nM -
CHEMBL2170307 Ki > 10000.0 nM -
CHEMBL2170306 Ki > 10000.0 nM -
CHEMBL2170305 Ki > 10000.0 nM -
CHEMBL1783426 Ki > 10000.0 nM -
CHEMBL2170304 Ki > 10000.0 nM -
CHEMBL2170315 Ki > 10000.0 nM -