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Assay Detail

CHEMBL2208708

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against respiratory syncytial virus
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Respiratory syncytial virus
Confidence 1 — Organism
Curated By Autocuration

Target

Respiratory syncytial virus (CHEMBL612679)
Type ORGANISM
Organism Respiratory syncytial virus

Publication

Synopsis of some recent tactical application of bioisosteres in drug design.
Meanwell NA.
J Med Chem (2011) 54 : 2529 -2591
PubMed 21413808 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 9 7.78 8.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL234027 1 8.52
CHEMBL233892 1 8.52
CHEMBL233786 1 8.52
CHEMBL446708 1 8.40
CHEMBL14710 1 8.30
CHEMBL388039 1 8.00
CHEMBL233893 1 7.80
CHEMBL392781 1 6.70
CHEMBL2203633 1 5.24

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL234027 EC50 = 3.0 nM 8.52
CHEMBL233892 EC50 = 3.0 nM 8.52
CHEMBL233786 EC50 = 3.0 nM 8.52
CHEMBL446708 EC50 = 4.0 nM 8.40
CHEMBL14710 EC50 = 5.0 nM 8.30
CHEMBL388039 EC50 = 10.0 nM 8.00
CHEMBL233893 EC50 = 16.0 nM 7.80
CHEMBL392781 EC50 = 200.0 nM 6.70
CHEMBL2203633 EC50 = 5700.0 nM 5.24