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Assay Detail

CHEMBL2210778

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of growth in TSC2-deficient MEF cells after 6 days
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type MEF
Confidence 1 — Organism
Curated By Autocuration

Target

MEF (CHEMBL614342)
Type CELL-LINE
Organism Mus musculus

Publication

Natural product-derived antitumor compound phenethyl isothiocyanate inhibits mTORC1 activity via TSC2.
Cavell BE, Syed Alwi SS, Donlevy AM, Proud CG, Packham G.
J Nat Prod (2012) 75 : 1051 -1057
PubMed 22607231 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.10 5.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL151649 PHENETHYLISOTHIOCYANATE 1 5.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL151649 PHENETHYLISOTHIOCYANATE IC50 = 8000.0 nM 5.10