Assay Detail
Functional
CHEMBL2214303
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against vincristine-resistant human HL60/Vinc cells incubated for 72 hrs by MTT assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Antiproliferative activity of salinomycin and its derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 5.23 | 6.04 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.04 |
| CHEMBL1208572 | SALINOMYCIN | 2.0 | 1 | 5.46 |
| CHEMBL2047977 | — | — | 1 | 5.37 |
| CHEMBL2047973 | — | — | 1 | 5.37 |
| CHEMBL2207532 | — | — | 1 | 5.28 |
| CHEMBL2047974 | — | — | 1 | 5.28 |
| CHEMBL2047976 | — | — | 1 | 5.22 |
| CHEMBL2207533 | — | — | 1 | 5.16 |
| CHEMBL2207534 | — | — | 1 | 4.55 |
| CHEMBL2047978 | — | — | 1 | 4.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 910.0 | nM | 6.04 |
| CHEMBL1208572 | SALINOMYCIN | IC50 | = | 3440.0 | nM | 5.46 |
| CHEMBL2047977 | — | IC50 | = | 4310.0 | nM | 5.37 |
| CHEMBL2047973 | — | IC50 | = | 4310.0 | nM | 5.37 |
| CHEMBL2207532 | — | IC50 | = | 5250.0 | nM | 5.28 |
| CHEMBL2047974 | — | IC50 | = | 5310.0 | nM | 5.28 |
| CHEMBL2047976 | — | IC50 | = | 6020.0 | nM | 5.22 |
| CHEMBL2207533 | — | IC50 | = | 6870.0 | nM | 5.16 |
| CHEMBL2207534 | — | IC50 | = | 28080.0 | nM | 4.55 |
| CHEMBL2047978 | — | IC50 | = | 29110.0 | nM | 4.54 |