Assay Detail
Functional
CHEMBL2214304
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human HL60 cells incubated for 72 hrs by MTT assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HL-60 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Antiproliferative activity of salinomycin and its derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 5.64 | 7.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.22 |
| CHEMBL1208572 | SALINOMYCIN | 2.0 | 1 | 6.36 |
| CHEMBL2207532 | — | — | 1 | 5.74 |
| CHEMBL2207533 | — | — | 1 | 5.51 |
| CHEMBL2047977 | — | — | 1 | 5.45 |
| CHEMBL2047976 | — | — | 1 | 5.44 |
| CHEMBL2047973 | — | — | 1 | 5.42 |
| CHEMBL2047974 | — | — | 1 | 5.41 |
| CHEMBL2207534 | — | — | 1 | 5.25 |
| CHEMBL2047978 | — | — | 1 | 4.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL1208572 | SALINOMYCIN | IC50 | = | 440.0 | nM | 6.36 |
| CHEMBL2207532 | — | IC50 | = | 1840.0 | nM | 5.74 |
| CHEMBL2207533 | — | IC50 | = | 3080.0 | nM | 5.51 |
| CHEMBL2047977 | — | IC50 | = | 3520.0 | nM | 5.45 |
| CHEMBL2047976 | — | IC50 | = | 3630.0 | nM | 5.44 |
| CHEMBL2047973 | — | IC50 | = | 3790.0 | nM | 5.42 |
| CHEMBL2047974 | — | IC50 | = | 3880.0 | nM | 5.41 |
| CHEMBL2207534 | — | IC50 | = | 5630.0 | nM | 5.25 |
| CHEMBL2047978 | — | IC50 | = | 24880.0 | nM | 4.60 |