Assay Detail
Functional
CHEMBL2214342
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at androgen receptor by cellular reporter gene assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Novel progesterone receptor modulators: 4-aryl-phenylsulfonamides.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.53 | 8.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL267431 | ASOPRISNIL | 3.0 | 1 | 8.05 |
| CHEMBL2203836 | — | — | 1 | 7.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL267431 | ASOPRISNIL | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL2203836 | — | IC50 | = | 100.0 | nM | 7.00 |