Assay Detail
Binding
CHEMBL2320213
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of urinary kallikrein (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development of new cyclic plasmin inhibitors with excellent potency and selectivity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.00 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2315243 | — | — | 1 | 5.00 |
| CHEMBL2315239 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2315243 | — | Ki | = | 10000.0 | nM | 5.00 |
| CHEMBL2315239 | — | Ki | > | 50000.0 | nM | - |