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Assay Detail

CHEMBL2320856

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Machupo virus
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mammarenavirus machupoense
Confidence 1 — Organism
Curated By Autocuration

Target

Machupo mammarenavirus (CHEMBL4888477)
Type ORGANISM
Organism Mammarenavirus machupoense

Publication

Discovery and optimization of potent broad-spectrum arenavirus inhibitors derived from benzimidazole and related heterocycles.
Burgeson JR, Moore AL, Gharaibeh DN, Larson RA, Cerruti NR, Amberg SM, Hruby DE, Dai D.
Bioorg Med Chem Lett (2013) 23 : 750 -756
PubMed 23265900 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 7.64 8.51

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2314859 1 8.51
CHEMBL2315146 1 7.55
CHEMBL2315140 1 7.40
CHEMBL2315147 1 7.09

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2314859 EC50 = 3.1 nM 8.51
CHEMBL2315146 EC50 = 28.0 nM 7.55
CHEMBL2315140 EC50 = 40.0 nM 7.40
CHEMBL2315147 EC50 = 81.0 nM 7.09