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Assay Detail

CHEMBL2327385

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Functional
Antiangiogenic activity in HMVEC assessed as inhibition of endothelial cell migration after 4 hrs by stereomicroscopic analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type Endothelial cell
Confidence 1 — Organism
Curated By Autocuration

Publication

1,2,3,4,6-Penta-O-galloyl-β-D-glucopyranose inhibits angiogenesis via inhibition of capillary morphogenesis gene 2.
Cryan LM, Bazinet L, Habeshian KA, Cao S, Clardy J, Christensen KA, Rogers MS.
J Med Chem (2013) 56 : 1940 -1945
PubMed 23394144 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.09 6.09

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL382408 PENTAGALLOYL GLUCOSE 1 6.09

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL382408 PENTAGALLOYL GLUCOSE IC50 = 820.0 nM 6.09