Assay Detail
Binding
CHEMBL2328683
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]Nalpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK-293 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Bodilisant-a novel fluorescent, highly affine histamine h3 receptor ligand.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.77 | 8.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2323582 | BODILISANT | — | 1 | 8.19 |
| CHEMBL14638 | CIPROXIFAN | — | 1 | 7.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2323582 | BODILISANT | Ki | = | 6.51 | nM | 8.19 |
| CHEMBL14638 | CIPROXIFAN | Ki | = | 46.0 | nM | 7.34 |