Assay Detail
Binding
CHEMBL2329795
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Inhibition of tPMET complex in human HL60 cells after 30 mins by WST-1/mPMS reduction assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HL-60 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Anti-leukemic activity of ubiquinone-based compounds targeting trans-plasma membrane electron transport.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 4.70 | 5.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2323207 | — | — | 1 | 5.22 |
| CHEMBL2323214 | — | — | 1 | 5.05 |
| CHEMBL2323215 | — | — | 1 | 5.00 |
| CHEMBL2323216 | — | — | 1 | 4.85 |
| CHEMBL2323209 | — | — | 1 | 4.85 |
| CHEMBL2323208 | — | — | 1 | 4.68 |
| CHEMBL2323212 | — | — | 1 | 4.64 |
| CHEMBL2323210 | — | — | 1 | 4.48 |
| CHEMBL252556 | IDEBENONE | 4.0 | 1 | 4.11 |
| CHEMBL2323206 | — | — | 1 | 4.09 |
| CHEMBL2323213 | — | — | 1 | - |
| CHEMBL2323211 | — | — | 1 | - |
| CHEMBL2323205 | — | — | 1 | - |
| CHEMBL2323204 | — | — | 1 | - |
| CHEMBL2323217 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2323207 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL2323214 | — | IC50 | = | 9000.0 | nM | 5.05 |
| CHEMBL2323215 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL2323216 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL2323209 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL2323208 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL2323212 | — | IC50 | = | 23000.0 | nM | 4.64 |
| CHEMBL2323210 | — | IC50 | = | 33000.0 | nM | 4.48 |
| CHEMBL252556 | IDEBENONE | IC50 | = | 77000.0 | nM | 4.11 |
| CHEMBL2323206 | — | IC50 | = | 81000.0 | nM | 4.09 |
| CHEMBL2323213 | — | IC50 | = | 122000.0 | nM | - |
| CHEMBL2323211 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL2323205 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL2323204 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL2323217 | — | IC50 | > | 200000.0 | nM | - |