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Compound Detail

CHEMBL2323211

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COC1=C(OC)C(=O)C(CCCCCCCCCCN(Cc2ccccc2)Cc2ccccc2)=C(C)C1=O

Basic Information

ChEMBL ID CHEMBL2323211
Phase Preclinical
Structure Type MOL
InChI Key NDIDZGLVGFJXNQ-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

517.7
MW (Da)
7.17
ALogP
5
HBA
0
HBD
55.8
PSA (Ų)
0.16
QED
2
Ro5 Violations
17
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C33H43NO4
MW 517.71
Aromatic Rings 2
Heavy Atoms 38
NP-Likeness 0.31

Activity Summary

IC50 1 meas. best 4.48

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
HL-60
CHEMBL383
IC50 4.48 4.48 33000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
HL-60 IC50 = 33000.0 nM 4.48 Antiproliferative activity against human HL60 cells after 48 hrs by MTT assay 23432053

Literature References

PubMed DOI Target Context # Activities
23432053 10.1021/jm301585z HL-60 2
23432053 10.1021/jm301585z Unchecked 2

Data from ChEMBL 36 via Core Engine