Assay Detail
Functional
CHEMBL2329763
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Antiproliferative activity against human HL60 cells after 48 hrs by MTT assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HL-60 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Anti-leukemic activity of ubiquinone-based compounds targeting trans-plasma membrane electron transport.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 5.16 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2323213 | — | — | 1 | 6.00 |
| CHEMBL2323216 | — | — | 1 | 5.70 |
| CHEMBL2323214 | — | — | 1 | 5.70 |
| CHEMBL2323215 | — | — | 1 | 5.52 |
| CHEMBL2323210 | — | — | 1 | 5.52 |
| CHEMBL2323209 | — | — | 1 | 5.52 |
| CHEMBL2323204 | — | — | 1 | 4.89 |
| CHEMBL2323217 | — | — | 1 | 4.89 |
| CHEMBL2323207 | — | — | 1 | 4.80 |
| CHEMBL2323211 | — | — | 1 | 4.48 |
| CHEMBL2323212 | — | — | 1 | 4.46 |
| CHEMBL252556 | IDEBENONE | 4.0 | 1 | 4.44 |
| CHEMBL2323208 | — | — | 1 | - |
| CHEMBL2323206 | — | — | 1 | - |
| CHEMBL2323205 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2323213 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL2323216 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL2323214 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL2323215 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL2323210 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL2323209 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL2323204 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL2323217 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL2323207 | — | IC50 | = | 16000.0 | nM | 4.80 |
| CHEMBL2323211 | — | IC50 | = | 33000.0 | nM | 4.48 |
| CHEMBL2323212 | — | IC50 | = | 35000.0 | nM | 4.46 |
| CHEMBL252556 | IDEBENONE | IC50 | = | 36000.0 | nM | 4.44 |
| CHEMBL2323208 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL2323206 | — | IC50 | = | 143000.0 | nM | - |
| CHEMBL2323205 | — | IC50 | > | 200000.0 | nM | - |