Assay Detail
Binding
CHEMBL2330915
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Inhibition of PKC delta (unknown origin) using ERMRPRKRQGSVRRRV as substrate after 15 mins by spectrophotometry in presence of ATP
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Design and optimization of selective protein kinase C θ (PKCθ) inhibitors for the treatment of autoimmune diseases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 27 | 6.75 | 7.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2326002 | — | — | 1 | 7.80 |
| CHEMBL2326001 | — | — | 1 | 7.75 |
| CHEMBL2326007 | — | — | 1 | 7.24 |
| CHEMBL2046626 | — | — | 1 | 7.10 |
| CHEMBL2326016 | — | — | 1 | 7.09 |
| CHEMBL2326019 | — | — | 1 | 7.05 |
| CHEMBL2326009 | — | — | 1 | 6.92 |
| CHEMBL2326004 | — | — | 1 | 6.89 |
| CHEMBL2326017 | — | — | 1 | 6.88 |
| CHEMBL2326018 | — | — | 1 | 6.88 |
| CHEMBL2326020 | — | — | 1 | 6.82 |
| CHEMBL2325999 | — | — | 1 | 6.62 |
| CHEMBL2046624 | — | — | 1 | 6.59 |
| CHEMBL2321918 | — | — | 1 | 6.47 |
| CHEMBL2326003 | — | — | 1 | 6.45 |
| CHEMBL2326011 | — | — | 1 | 6.32 |
| CHEMBL2326014 | — | — | 1 | 6.28 |
| CHEMBL2326012 | — | — | 1 | 6.26 |
| CHEMBL2326015 | — | — | 1 | 6.14 |
| CHEMBL2326021 | — | — | 1 | 6.10 |
| CHEMBL2326013 | — | — | 1 | 6.02 |
| CHEMBL2326005 | — | — | 1 | - |
| CHEMBL2326006 | — | — | 1 | - |
| CHEMBL2326008 | — | — | 1 | - |
| CHEMBL2326010 | — | — | 1 | - |
| CHEMBL2325998 | — | — | 1 | - |
| CHEMBL2326000 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2326002 | — | Ki | = | 16.0 | nM | 7.80 |
| CHEMBL2326001 | — | Ki | = | 18.0 | nM | 7.75 |
| CHEMBL2326007 | — | Ki | = | 57.0 | nM | 7.24 |
| CHEMBL2046626 | — | Ki | = | 80.0 | nM | 7.10 |
| CHEMBL2326016 | — | Ki | = | 81.0 | nM | 7.09 |
| CHEMBL2326019 | — | Ki | = | 89.0 | nM | 7.05 |
| CHEMBL2326009 | — | Ki | = | 120.0 | nM | 6.92 |
| CHEMBL2326004 | — | Ki | = | 130.0 | nM | 6.89 |
| CHEMBL2326017 | — | Ki | = | 132.0 | nM | 6.88 |
| CHEMBL2326018 | — | Ki | = | 131.0 | nM | 6.88 |
| CHEMBL2326020 | — | Ki | = | 151.0 | nM | 6.82 |
| CHEMBL2325999 | — | Ki | = | 242.0 | nM | 6.62 |
| CHEMBL2046624 | — | Ki | = | 255.0 | nM | 6.59 |
| CHEMBL2321918 | — | Ki | = | 336.0 | nM | 6.47 |
| CHEMBL2326003 | — | Ki | = | 358.0 | nM | 6.45 |
| CHEMBL2326011 | — | Ki | = | 480.0 | nM | 6.32 |
| CHEMBL2326014 | — | Ki | = | 526.0 | nM | 6.28 |
| CHEMBL2326012 | — | Ki | = | 547.0 | nM | 6.26 |
| CHEMBL2326015 | — | Ki | = | 722.0 | nM | 6.14 |
| CHEMBL2326021 | — | Ki | = | 792.0 | nM | 6.10 |
| CHEMBL2326013 | — | Ki | = | 957.0 | nM | 6.02 |
| CHEMBL2326005 | — | Ki | > | 1250.0 | nM | - |
| CHEMBL2326006 | — | Ki | > | 1250.0 | nM | - |
| CHEMBL2326008 | — | Ki | > | 1250.0 | nM | - |
| CHEMBL2326010 | — | Ki | > | 1250.0 | nM | - |
| CHEMBL2325998 | — | Ki | < | 10.0 | nM | - |
| CHEMBL2326000 | — | Ki | < | 10.0 | nM | - |