Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL2339946

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Activation of Staphylococcus aureus AgrC1
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Staphylococcus aureus
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

ADMET (CHEMBL612558)
Type ADMET

Publication

Attenuating Staphylococcus aureus virulence gene regulation: a medicinal chemistry perspective.
Gordon CP, Williams P, Chan WC.
J Med Chem (2013) 56 : 1389 -1404
PubMed 23294220 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 6.40 7.55

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2337554 1 7.55
CHEMBL2337556 1 5.24

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2337554 EC50 = 28.0 nM 7.55
CHEMBL2337556 EC50 = 5800.0 nM 5.24