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Assay Detail

CHEMBL2340978

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of AChE (unknown origin)
3
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Acetylcholinesterase (CHEMBL220)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Structural analogs of huperzine A improve survival in guinea pigs exposed to soman.
Gunosewoyo H, Tipparaju SK, Pieroni M, Wang Y, Doctor BP, Nambiar MP, Kozikowski AP.
Bioorg Med Chem Lett (2013) 23 : 1544 -1547
PubMed 23395652 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
INH 2 - -
IC50 1 7.35 7.35

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL395280 HUPERZINE A 2.0 1 7.35
CHEMBL2333849 1 -
CHEMBL2333848 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL395280 HUPERZINE A IC50 = 45.0 nM 7.35
CHEMBL2333849 INH = 10.0 uM -
CHEMBL2333848 INH = 5.0 uM -