Assay Detail
Binding
CHEMBL2350427
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Inhibition of c-MET phosphorylation (unknown origin) after 1 hr by Z'-LYTE kinase assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Olive secoiridoids and semisynthetic bioisostere analogues for the control of metastatic breast cancer.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.06 | 5.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2172394 | (-)-OLEOCANTHAL | — | 1 | 5.26 |
| CHEMBL2348314 | TYROSOL SINAPATE | — | 1 | 4.86 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2172394 | (-)-OLEOCANTHAL | IC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL2348314 | TYROSOL SINAPATE | IC50 | = | 13700.0 | nM | 4.86 |