Assay Detail
Functional
CHEMBL2363142
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SANGER: Inhibition of human COLO-829 cell growth in a cell viability assay.
136
Total Activities
134
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | COLO-829 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 136 | 5.44 | 9.98 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 9.98 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.21 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.14 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.93 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.72 |
| CHEMBL2144069 | — | — | 1 | 7.59 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.53 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.49 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.37 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.92 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 6.91 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.71 |
| CHEMBL1256459 | TORIN1 | — | 1 | 6.68 |
| CHEMBL64925 | MG-132 | — | 2 | 6.62 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.53 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.53 |
| CHEMBL213100 | — | — | 1 | 6.51 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 6.46 |
| CHEMBL1230020 | PLX-4720 | — | 1 | 6.41 |
| CHEMBL585951 | — | — | 1 | 6.28 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 6.24 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.18 |
| CHEMBL217354 | — | — | 1 | 6.16 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.14 |
| CHEMBL1084546 | PF-00562271 | 1.0 | 1 | 6.12 |
| CHEMBL2363137 | — | — | 1 | 6.08 |
| CHEMBL477989 | SB590885 | — | 1 | 6.01 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.93 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 5.89 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 5.84 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL553025 | VINORELBINE | IC50 | = | 0.1051 | nM | 9.98 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.6136 | nM | 9.21 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 7.248 | nM | 8.14 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 11.67 | nM | 7.93 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 19.17 | nM | 7.72 |
| CHEMBL2144069 | — | IC50 | = | 25.65 | nM | 7.59 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 29.82 | nM | 7.53 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 32.15 | nM | 7.49 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 43.11 | nM | 7.37 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 120.05 | nM | 6.92 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 122.13 | nM | 6.91 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 196.77 | nM | 6.71 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 206.73 | nM | 6.68 |
| CHEMBL64925 | MG-132 | IC50 | = | 242.57 | nM | 6.62 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 298.45 | nM | 6.53 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 296.5 | nM | 6.53 |
| CHEMBL213100 | — | IC50 | = | 312.12 | nM | 6.51 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 344.52 | nM | 6.46 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 389.68 | nM | 6.41 |
| CHEMBL585951 | — | IC50 | = | 520.1 | nM | 6.28 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 575.7 | nM | 6.24 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 657.99 | nM | 6.18 |
| CHEMBL217354 | — | IC50 | = | 700.55 | nM | 6.16 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 719.85 | nM | 6.14 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 751.76 | nM | 6.12 |
| CHEMBL2363137 | — | IC50 | = | 824.54 | nM | 6.08 |
| CHEMBL477989 | SB590885 | IC50 | = | 966.94 | nM | 6.01 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1161.06 | nM | 5.93 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 1274.87 | nM | 5.89 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 1429.79 | nM | 5.84 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1535.64 | nM | 5.81 |
| CHEMBL105442 | CI-1040 | IC50 | = | 1622.32 | nM | 5.79 |
| CHEMBL3349342 | — | IC50 | = | 1730.77 | nM | 5.76 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1768.57 | nM | 5.75 |
| CHEMBL803 | CYTARABINE | IC50 | = | 1864.71 | nM | 5.73 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 2086.84 | nM | 5.68 |
| CHEMBL379975 | — | IC50 | = | 2186.49 | nM | 5.66 |
| CHEMBL202721 | — | IC50 | = | 2639.0 | nM | 5.58 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 2765.4 | nM | 5.56 |
| CHEMBL135561 | — | IC50 | = | 2951.95 | nM | 5.53 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 3242.26 | nM | 5.49 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 3500.73 | nM | 5.46 |
| CHEMBL573107 | — | IC50 | = | 3666.18 | nM | 5.44 |
| CHEMBL300389 | — | IC50 | = | 4176.22 | nM | 5.38 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 4134.6 | nM | 5.38 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 4770.43 | nM | 5.32 |
| CHEMBL221137 | EMBELIN | IC50 | = | 5290.16 | nM | 5.28 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 5498.84 | nM | 5.26 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 5915.04 | nM | 5.23 |
| CHEMBL514499 | GW843682X | IC50 | = | 6263.86 | nM | 5.20 |