Assay Detail
Functional
CHEMBL2363156
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human Ca9-22 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Ca9-22 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.83 | 9.37 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.37 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.95 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.81 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.65 |
| CHEMBL217354 | — | — | 1 | 8.42 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.37 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.19 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.99 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.64 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.55 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.47 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.30 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 7.08 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.01 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.95 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.81 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.72 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.49 |
| CHEMBL585951 | — | — | 1 | 6.41 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.30 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.27 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.24 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.23 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.13 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.10 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.05 |
| CHEMBL3349342 | — | — | 1 | 6.01 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 5.98 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 5.81 |
| CHEMBL577784 | BX-795 | — | 1 | 5.67 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.4234 | nM | 9.37 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 1.131 | nM | 8.95 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 1.538 | nM | 8.81 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 2.211 | nM | 8.65 |
| CHEMBL217354 | — | IC50 | = | 3.82 | nM | 8.42 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 4.247 | nM | 8.37 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 6.391 | nM | 8.19 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 10.27 | nM | 7.99 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 22.78 | nM | 7.64 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 27.96 | nM | 7.55 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 33.55 | nM | 7.47 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 50.07 | nM | 7.30 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 83.53 | nM | 7.08 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 96.61 | nM | 7.01 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 111.28 | nM | 6.95 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 155.57 | nM | 6.81 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 190.35 | nM | 6.72 |
| CHEMBL803 | CYTARABINE | IC50 | = | 320.77 | nM | 6.49 |
| CHEMBL585951 | — | IC50 | = | 389.48 | nM | 6.41 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 504.94 | nM | 6.30 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 540.77 | nM | 6.27 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 580.63 | nM | 6.24 |
| CHEMBL939 | GEFITINIB | IC50 | = | 588.64 | nM | 6.23 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 745.83 | nM | 6.13 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 787.36 | nM | 6.10 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 899.91 | nM | 6.05 |
| CHEMBL3349342 | — | IC50 | = | 981.15 | nM | 6.01 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 1051.07 | nM | 5.98 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 1562.6 | nM | 5.81 |
| CHEMBL577784 | BX-795 | IC50 | = | 2128.47 | nM | 5.67 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 2188.07 | nM | 5.66 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 2376.67 | nM | 5.62 |
| CHEMBL135561 | — | IC50 | = | 2614.63 | nM | 5.58 |
| CHEMBL573107 | — | IC50 | = | 2659.33 | nM | 5.58 |
| CHEMBL379975 | — | IC50 | = | 2896.88 | nM | 5.54 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 2937.67 | nM | 5.53 |
| CHEMBL105442 | CI-1040 | IC50 | = | 2972.55 | nM | 5.53 |
| CHEMBL202721 | — | IC50 | = | 3289.6 | nM | 5.48 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 3404.94 | nM | 5.47 |
| CHEMBL399530 | — | IC50 | = | 4281.57 | nM | 5.37 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 4456.91 | nM | 5.35 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 4555.16 | nM | 5.34 |
| CHEMBL2363137 | — | IC50 | = | 5998.74 | nM | 5.22 |
| CHEMBL258844 | — | IC50 | = | 5973.33 | nM | 5.22 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 6167.1 | nM | 5.21 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 6690.8 | nM | 5.17 |
| CHEMBL512504 | — | IC50 | = | 8627.48 | nM | 5.06 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 9328.75 | nM | 5.03 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 10066.53 | nM | 5.00 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 10391.9 | nM | 4.98 |