Assay Detail
Functional
CHEMBL2363171
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SANGER: Inhibition of human D-502MG cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | D-502MG |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.30 | 8.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.39 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.20 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.78 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.65 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.63 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.59 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.08 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.98 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 6.96 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.62 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.46 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.39 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 6.32 |
| CHEMBL2363137 | — | — | 1 | 6.22 |
| CHEMBL585951 | — | — | 1 | 5.98 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 5.91 |
| CHEMBL64925 | MG-132 | — | 2 | 5.78 |
| CHEMBL300389 | — | — | 1 | 5.73 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 5.72 |
| CHEMBL2144069 | — | — | 1 | 5.65 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 5.63 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 5.57 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 5.54 |
| CHEMBL191334 | NUTLIN-3 | — | 1 | 5.53 |
| CHEMBL573107 | — | — | 1 | 5.51 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 5.50 |
| CHEMBL379300 | A-443654 | — | 1 | 5.48 |
| CHEMBL3349342 | — | — | 1 | 5.42 |
| CHEMBL202721 | — | — | 1 | 5.40 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 5.38 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 4.102 | nM | 8.39 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 6.375 | nM | 8.20 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 16.72 | nM | 7.78 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 22.59 | nM | 7.65 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 23.49 | nM | 7.63 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 25.81 | nM | 7.59 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 82.63 | nM | 7.08 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 105.7 | nM | 6.98 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 111.01 | nM | 6.96 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 241.74 | nM | 6.62 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 343.18 | nM | 6.46 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 411.27 | nM | 6.39 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 480.3 | nM | 6.32 |
| CHEMBL2363137 | — | IC50 | = | 606.81 | nM | 6.22 |
| CHEMBL585951 | — | IC50 | = | 1048.93 | nM | 5.98 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 1233.76 | nM | 5.91 |
| CHEMBL64925 | MG-132 | IC50 | = | 1672.11 | nM | 5.78 |
| CHEMBL300389 | — | IC50 | = | 1857.04 | nM | 5.73 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 1911.32 | nM | 5.72 |
| CHEMBL2144069 | — | IC50 | = | 2261.42 | nM | 5.65 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 2324.61 | nM | 5.63 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 2704.06 | nM | 5.57 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 2868.05 | nM | 5.54 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 2971.54 | nM | 5.53 |
| CHEMBL573107 | — | IC50 | = | 3070.19 | nM | 5.51 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 3143.9 | nM | 5.50 |
| CHEMBL379300 | A-443654 | IC50 | = | 3279.65 | nM | 5.48 |
| CHEMBL3349342 | — | IC50 | = | 3810.67 | nM | 5.42 |
| CHEMBL202721 | — | IC50 | = | 3969.79 | nM | 5.40 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 4169.97 | nM | 5.38 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 4365.48 | nM | 5.36 |
| CHEMBL217354 | — | IC50 | = | 4922.02 | nM | 5.31 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 5004.16 | nM | 5.30 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 5242.62 | nM | 5.28 |
| CHEMBL803 | CYTARABINE | IC50 | = | 5490.75 | nM | 5.26 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 5842.31 | nM | 5.23 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 6176.59 | nM | 5.21 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 6173.36 | nM | 5.21 |
| CHEMBL577784 | BX-795 | IC50 | = | 6270.74 | nM | 5.20 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 6288.57 | nM | 5.20 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 6320.47 | nM | 5.20 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 6423.76 | nM | 5.19 |
| CHEMBL554 | LAPATINIB | IC50 | = | 7488.94 | nM | 5.13 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 7384.73 | nM | 5.13 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 7782.22 | nM | 5.11 |
| CHEMBL513909 | BI-2536 | IC50 | = | 7983.6 | nM | 5.10 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 8292.82 | nM | 5.08 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 8534.92 | nM | 5.07 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 8786.29 | nM | 5.06 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 8769.94 | nM | 5.06 |