Assay Detail
Functional
CHEMBL2363176
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SANGER: Inhibition of human DEL cell growth in a cell viability assay.
130
Total Activities
129
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | DEL |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 130 | 5.85 | 10.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 10.05 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.09 |
| CHEMBL509032 | TAE-684 | — | 1 | 9.03 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.67 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.52 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 8.51 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.44 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.37 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 8.26 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.07 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.99 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 7.75 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.72 |
| CHEMBL514499 | GW843682X | — | 1 | 7.70 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.69 |
| CHEMBL300389 | — | — | 1 | 7.59 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.55 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.42 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 7.34 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 7.33 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.32 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.24 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.08 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 6.95 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.81 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.73 |
| CHEMBL379300 | A-443654 | — | 1 | 6.64 |
| CHEMBL512504 | — | — | 1 | 6.64 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.57 |
| CHEMBL585951 | — | — | 1 | 6.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.08871 | nM | 10.05 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.8157 | nM | 9.09 |
| CHEMBL509032 | TAE-684 | IC50 | = | 0.9269 | nM | 9.03 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 2.16 | nM | 8.67 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 3.012 | nM | 8.52 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 3.119 | nM | 8.51 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 3.63 | nM | 8.44 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 4.293 | nM | 8.37 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 5.46 | nM | 8.26 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 8.449 | nM | 8.07 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 10.34 | nM | 7.99 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 17.99 | nM | 7.75 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 19.22 | nM | 7.72 |
| CHEMBL514499 | GW843682X | IC50 | = | 19.94 | nM | 7.70 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 20.49 | nM | 7.69 |
| CHEMBL300389 | — | IC50 | = | 25.84 | nM | 7.59 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 28.15 | nM | 7.55 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 38.44 | nM | 7.42 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 45.92 | nM | 7.34 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 47.28 | nM | 7.33 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 48.39 | nM | 7.32 |
| CHEMBL513909 | BI-2536 | IC50 | = | 57.09 | nM | 7.24 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 83.47 | nM | 7.08 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 111.92 | nM | 6.95 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 153.81 | nM | 6.81 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 184.5 | nM | 6.73 |
| CHEMBL379300 | A-443654 | IC50 | = | 231.45 | nM | 6.64 |
| CHEMBL512504 | — | IC50 | = | 228.25 | nM | 6.64 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 270.65 | nM | 6.57 |
| CHEMBL585951 | — | IC50 | = | 288.8 | nM | 6.54 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 311.49 | nM | 6.51 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 374.87 | nM | 6.43 |
| CHEMBL601719 | CRIZOTINIB | IC50 | = | 369.9 | nM | 6.43 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 391.27 | nM | 6.41 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 479.88 | nM | 6.32 |
| CHEMBL379975 | — | IC50 | = | 485.03 | nM | 6.31 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 558.98 | nM | 6.25 |
| CHEMBL803 | CYTARABINE | IC50 | = | 874.85 | nM | 6.06 |
| CHEMBL939 | GEFITINIB | IC50 | = | 877.65 | nM | 6.06 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 967.73 | nM | 6.01 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1025.9 | nM | 5.99 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1100.05 | nM | 5.96 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 1256.43 | nM | 5.90 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 1254.57 | nM | 5.90 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 1351.62 | nM | 5.87 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 1409.39 | nM | 5.85 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 1436.57 | nM | 5.84 |
| CHEMBL64925 | MG-132 | IC50 | = | 1592.1 | nM | 5.80 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1702.73 | nM | 5.77 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 1746.92 | nM | 5.76 |