Assay Detail
Functional
CHEMBL2363191
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SANGER: Inhibition of human Daoy cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Daoy |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.82 | 10.56 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 10.56 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 9.34 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.32 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.15 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.51 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.27 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.18 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 8.16 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 8.09 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.78 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.43 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.29 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.25 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 7.24 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.23 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 7.08 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.05 |
| CHEMBL217354 | — | — | 1 | 6.85 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.80 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.50 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.43 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.35 |
| CHEMBL558642 | GSK-650394 | — | 1 | 6.29 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.27 |
| CHEMBL585951 | — | — | 1 | 6.06 |
| CHEMBL573107 | — | — | 1 | 6.00 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.98 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.96 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.92 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 5.87 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.02733 | nM | 10.56 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.4565 | nM | 9.34 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.4809 | nM | 9.32 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.7004 | nM | 9.15 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 3.102 | nM | 8.51 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 5.343 | nM | 8.27 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 6.646 | nM | 8.18 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 6.953 | nM | 8.16 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 8.073 | nM | 8.09 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 16.8 | nM | 7.78 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 36.7 | nM | 7.43 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 51.72 | nM | 7.29 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 56.16 | nM | 7.25 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 57.53 | nM | 7.24 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 58.64 | nM | 7.23 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 83.04 | nM | 7.08 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 88.01 | nM | 7.05 |
| CHEMBL217354 | — | IC50 | = | 140.73 | nM | 6.85 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 158.77 | nM | 6.80 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 317.23 | nM | 6.50 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 367.73 | nM | 6.43 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 451.03 | nM | 6.35 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 515.32 | nM | 6.29 |
| CHEMBL803 | CYTARABINE | IC50 | = | 532.22 | nM | 6.27 |
| CHEMBL585951 | — | IC50 | = | 864.7 | nM | 6.06 |
| CHEMBL573107 | — | IC50 | = | 987.67 | nM | 6.00 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1044.6 | nM | 5.98 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1096.28 | nM | 5.96 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1208.48 | nM | 5.92 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 1335.7 | nM | 5.87 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 1507.37 | nM | 5.82 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 1763.19 | nM | 5.75 |
| CHEMBL591429 | PAC-1 | IC50 | = | 2185.64 | nM | 5.66 |
| CHEMBL379975 | — | IC50 | = | 2738.48 | nM | 5.56 |
| CHEMBL259181 | — | IC50 | = | 2930.43 | nM | 5.53 |
| CHEMBL472940 | — | IC50 | = | 3246.62 | nM | 5.49 |
| CHEMBL2363137 | — | IC50 | = | 4139.6 | nM | 5.38 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 4779.49 | nM | 5.32 |
| CHEMBL399530 | — | IC50 | = | 4924.54 | nM | 5.31 |
| CHEMBL577784 | BX-795 | IC50 | = | 5509.94 | nM | 5.26 |
| CHEMBL221137 | EMBELIN | IC50 | = | 5464.66 | nM | 5.26 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 5726.42 | nM | 5.24 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 7943.21 | nM | 5.10 |
| CHEMBL202721 | — | IC50 | = | 8959.16 | nM | 5.05 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 9120.28 | nM | 5.04 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 9241.43 | nM | 5.03 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 9357.4 | nM | 5.03 |
| CHEMBL191384 | — | IC50 | = | 9797.7 | nM | 5.01 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 10220.23 | nM | 4.99 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 11433.62 | nM | 4.94 |