Assay Detail
Functional
CHEMBL2363192
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SANGER: Inhibition of human Daudi cell growth in a cell viability assay.
78
Total Activities
77
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Daudi |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 78 | 5.89 | 9.36 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 9.36 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.91 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.44 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.77 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.61 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 7.60 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.47 |
| CHEMBL514499 | GW843682X | — | 1 | 7.46 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.37 |
| CHEMBL512504 | — | — | 1 | 7.30 |
| CHEMBL300389 | — | — | 1 | 7.26 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.16 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.15 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.08 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.07 |
| CHEMBL379300 | A-443654 | — | 1 | 6.45 |
| CHEMBL585951 | — | — | 1 | 6.42 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.41 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 6.25 |
| CHEMBL1190711 | — | — | 1 | 6.22 |
| CHEMBL213100 | — | — | 1 | 6.15 |
| CHEMBL27759 | ENTINOSTAT | 3.0 | 1 | 6.11 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.04 |
| CHEMBL591429 | PAC-1 | 1.0 | 1 | 6.02 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 1 | 5.97 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | — | 1 | 5.93 |
| CHEMBL2363137 | — | — | 1 | 5.90 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 5.78 |
| CHEMBL509032 | TAE-684 | — | 1 | 5.75 |
| CHEMBL64925 | MG-132 | — | 2 | 5.69 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL413 | SIROLIMUS | IC50 | = | 0.4336 | nM | 9.36 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 1.223 | nM | 8.91 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 3.633 | nM | 8.44 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 17.08 | nM | 7.77 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 24.77 | nM | 7.61 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 25.37 | nM | 7.60 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 33.76 | nM | 7.47 |
| CHEMBL514499 | GW843682X | IC50 | = | 34.68 | nM | 7.46 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 42.25 | nM | 7.37 |
| CHEMBL512504 | — | IC50 | = | 49.79 | nM | 7.30 |
| CHEMBL300389 | — | IC50 | = | 55.27 | nM | 7.26 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 68.96 | nM | 7.16 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 70.81 | nM | 7.15 |
| CHEMBL513909 | BI-2536 | IC50 | = | 82.56 | nM | 7.08 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 84.92 | nM | 7.07 |
| CHEMBL379300 | A-443654 | IC50 | = | 354.63 | nM | 6.45 |
| CHEMBL585951 | — | IC50 | = | 381.09 | nM | 6.42 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 392.42 | nM | 6.41 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 569.49 | nM | 6.25 |
| CHEMBL1190711 | — | IC50 | = | 606.99 | nM | 6.22 |
| CHEMBL213100 | — | IC50 | = | 714.11 | nM | 6.15 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 776.81 | nM | 6.11 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 921.4 | nM | 6.04 |
| CHEMBL591429 | PAC-1 | IC50 | = | 946.53 | nM | 6.02 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1068.88 | nM | 5.97 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 1173.2 | nM | 5.93 |
| CHEMBL2363137 | — | IC50 | = | 1251.97 | nM | 5.90 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 1670.96 | nM | 5.78 |
| CHEMBL509032 | TAE-684 | IC50 | = | 1789.67 | nM | 5.75 |
| CHEMBL64925 | MG-132 | IC50 | = | 2054.59 | nM | 5.69 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 2098.02 | nM | 5.68 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 2500.76 | nM | 5.60 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 3442.87 | nM | 5.46 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 3662.19 | nM | 5.44 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 5091.19 | nM | 5.29 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 5361.15 | nM | 5.27 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 5516.94 | nM | 5.26 |
| CHEMBL472940 | — | IC50 | = | 5684.77 | nM | 5.25 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 5691.2 | nM | 5.25 |
| CHEMBL221137 | EMBELIN | IC50 | = | 5749.14 | nM | 5.24 |
| CHEMBL180127 | SALUBRINAL | IC50 | = | 6336.99 | nM | 5.20 |
| CHEMBL197603 | — | IC50 | = | 6475.2 | nM | 5.19 |
| CHEMBL191384 | — | IC50 | = | 6540.61 | nM | 5.18 |
| CHEMBL535 | SUNITINIB | IC50 | = | 8235.46 | nM | 5.08 |
| CHEMBL258844 | — | IC50 | = | 10818.83 | nM | 4.97 |
| CHEMBL259181 | — | IC50 | = | 12851.7 | nM | 4.89 |
| CHEMBL1673039 | — | IC50 | = | 15478.41 | nM | 4.81 |
| CHEMBL1242367 | — | IC50 | = | 15760.79 | nM | 4.80 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 17614.93 | nM | 4.75 |
| CHEMBL64925 | MG-132 | IC50 | = | 18923.13 | nM | 4.72 |