Assay Detail
Functional
CHEMBL2363199
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SANGER: Inhibition of human ECC12 cell growth in a cell viability assay.
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | ECC12 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 29 | 5.72 | 9.29 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 9.29 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.86 |
| CHEMBL553 | ERLOTINIB | 4.0 | 1 | 7.09 |
| CHEMBL554 | LAPATINIB | 4.0 | 1 | 7.04 |
| CHEMBL585951 | — | — | 1 | 6.49 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.37 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.25 |
| CHEMBL27759 | ENTINOSTAT | 3.0 | 1 | 6.15 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.02 |
| CHEMBL2144069 | — | — | 1 | 5.77 |
| CHEMBL64925 | MG-132 | — | 1 | 5.62 |
| CHEMBL36 | PYRIMETHAMINE | 4.0 | 1 | 5.59 |
| CHEMBL1084546 | PF-00562271 | 1.0 | 1 | 5.11 |
| CHEMBL258844 | — | — | 1 | 5.05 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.02 |
| CHEMBL1673039 | — | — | 1 | 4.98 |
| CHEMBL135561 | — | — | 1 | 4.69 |
| CHEMBL1336 | SORAFENIB | 4.0 | 1 | 4.62 |
| CHEMBL512504 | — | — | 1 | 4.42 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 1 | 4.32 |
| CHEMBL180127 | SALUBRINAL | — | 1 | 4.31 |
| CHEMBL472004 | — | — | 1 | 4.23 |
| CHEMBL220241 | GSK-269962A | — | 1 | 4.22 |
| CHEMBL14762 | SELICICLIB | 2.0 | 1 | - |
| CHEMBL412142 | LADUVIGLUSIB | 1.0 | 1 | - |
| CHEMBL373751 | GSK-319347A | — | 1 | - |
| CHEMBL4298697 | — | — | 1 | - |
| CHEMBL92309 | — | — | 1 | - |
| CHEMBL254129 | CYCLOPAMINE | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL553025 | VINORELBINE | IC50 | = | 0.509 | nM | 9.29 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 1.373 | nM | 8.86 |
| CHEMBL553 | ERLOTINIB | IC50 | = | 80.52 | nM | 7.09 |
| CHEMBL554 | LAPATINIB | IC50 | = | 92.31 | nM | 7.04 |
| CHEMBL585951 | — | IC50 | = | 323.56 | nM | 6.49 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 429.23 | nM | 6.37 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 565.58 | nM | 6.25 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 700.86 | nM | 6.15 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 954.38 | nM | 6.02 |
| CHEMBL2144069 | — | IC50 | = | 1714.9 | nM | 5.77 |
| CHEMBL64925 | MG-132 | IC50 | = | 2379.4 | nM | 5.62 |
| CHEMBL36 | PYRIMETHAMINE | IC50 | = | 2561.76 | nM | 5.59 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 7729.01 | nM | 5.11 |
| CHEMBL258844 | — | IC50 | = | 8885.69 | nM | 5.05 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 9648.24 | nM | 5.02 |
| CHEMBL1673039 | — | IC50 | = | 10424.27 | nM | 4.98 |
| CHEMBL135561 | — | IC50 | = | 20489.67 | nM | 4.69 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 24280.27 | nM | 4.62 |
| CHEMBL512504 | — | IC50 | = | 37714.25 | nM | 4.42 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 47497.97 | nM | 4.32 |
| CHEMBL180127 | SALUBRINAL | IC50 | = | 48980.29 | nM | 4.31 |
| CHEMBL472004 | — | IC50 | = | 58692.44 | nM | 4.23 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 60482.92 | nM | 4.22 |
| CHEMBL14762 | SELICICLIB | IC50 | = | 288995.18 | nM | - |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 310253.59 | nM | - |
| CHEMBL373751 | GSK-319347A | IC50 | = | 375694.38 | nM | - |
| CHEMBL4298697 | — | IC50 | = | 158539.69 | nM | - |
| CHEMBL92309 | — | IC50 | = | 1796894.18 | nM | - |
| CHEMBL254129 | CYCLOPAMINE | IC50 | = | 753333.48 | nM | - |