Assay Detail
Functional
CHEMBL2363219
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human EVSA-T cell growth in a cell viability assay.
87
Total Activities
85
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | EVSA-T |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 87 | 5.44 | 8.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.44 |
| CHEMBL1256459 | TORIN1 | — | 1 | 8.05 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.51 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.41 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.03 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.92 |
| CHEMBL300389 | — | — | 1 | 6.87 |
| CHEMBL217354 | — | — | 1 | 6.85 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 6.69 |
| CHEMBL379300 | A-443654 | — | 1 | 6.66 |
| CHEMBL514499 | GW843682X | — | 1 | 6.62 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 6.56 |
| CHEMBL512504 | — | — | 1 | 6.42 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.39 |
| CHEMBL64925 | MG-132 | — | 2 | 6.30 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.18 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.09 |
| CHEMBL27759 | ENTINOSTAT | 3.0 | 1 | 5.93 |
| CHEMBL585951 | — | — | 1 | 5.90 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 5.80 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 5.66 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 5.64 |
| CHEMBL515416 | — | — | 1 | 5.62 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | — | 1 | 5.47 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 2 | 5.47 |
| CHEMBL554 | LAPATINIB | 4.0 | 1 | 5.13 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 5.03 |
| CHEMBL509032 | TAE-684 | — | 1 | 4.99 |
| CHEMBL217092 | SARACATINIB | 3.0 | 1 | 4.97 |
| CHEMBL1242367 | — | — | 1 | 4.97 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 3.599 | nM | 8.44 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 8.919 | nM | 8.05 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 30.73 | nM | 7.51 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 39.23 | nM | 7.41 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 92.65 | nM | 7.03 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 121.53 | nM | 6.92 |
| CHEMBL300389 | — | IC50 | = | 134.7 | nM | 6.87 |
| CHEMBL217354 | — | IC50 | = | 139.93 | nM | 6.85 |
| CHEMBL513909 | BI-2536 | IC50 | = | 203.12 | nM | 6.69 |
| CHEMBL379300 | A-443654 | IC50 | = | 220.18 | nM | 6.66 |
| CHEMBL514499 | GW843682X | IC50 | = | 236.88 | nM | 6.62 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 275.19 | nM | 6.56 |
| CHEMBL512504 | — | IC50 | = | 380.95 | nM | 6.42 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 409.8 | nM | 6.39 |
| CHEMBL64925 | MG-132 | IC50 | = | 499.11 | nM | 6.30 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 664.4 | nM | 6.18 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 816.72 | nM | 6.09 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1181.14 | nM | 5.93 |
| CHEMBL585951 | — | IC50 | = | 1265.91 | nM | 5.90 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 1573.68 | nM | 5.80 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 2173.15 | nM | 5.66 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 2300.89 | nM | 5.64 |
| CHEMBL515416 | — | IC50 | = | 2396.31 | nM | 5.62 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 3402.06 | nM | 5.47 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 3379.75 | nM | 5.47 |
| CHEMBL554 | LAPATINIB | IC50 | = | 7428.11 | nM | 5.13 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 9277.93 | nM | 5.03 |
| CHEMBL509032 | TAE-684 | IC50 | = | 10319.24 | nM | 4.99 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 10656.8 | nM | 4.97 |
| CHEMBL1242367 | — | IC50 | = | 10685.42 | nM | 4.97 |
| CHEMBL1673039 | — | IC50 | = | 10951.86 | nM | 4.96 |
| CHEMBL399530 | — | IC50 | = | 10894.16 | nM | 4.96 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 11960.88 | nM | 4.92 |
| CHEMBL2363137 | — | IC50 | = | 11908.82 | nM | 4.92 |
| CHEMBL180127 | SALUBRINAL | IC50 | = | 12920.39 | nM | 4.89 |
| CHEMBL209148 | — | IC50 | = | 14021.01 | nM | 4.85 |
| CHEMBL197603 | — | IC50 | = | 14203.37 | nM | 4.85 |
| CHEMBL213100 | — | IC50 | = | 15248.44 | nM | 4.82 |
| CHEMBL535 | SUNITINIB | IC50 | = | 17048.46 | nM | 4.77 |
| CHEMBL191384 | — | IC50 | = | 17345.24 | nM | 4.76 |
| CHEMBL401930 | — | IC50 | = | 17934.08 | nM | 4.75 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 20683.06 | nM | 4.68 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 21149.92 | nM | 4.67 |
| CHEMBL254129 | CYCLOPAMINE | IC50 | = | 27556.1 | nM | 4.56 |
| CHEMBL259181 | — | IC50 | = | 29566.38 | nM | 4.53 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 32258.51 | nM | 4.49 |
| CHEMBL64925 | MG-132 | IC50 | = | 40016.43 | nM | 4.40 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 42895.37 | nM | 4.37 |
| CHEMBL4298697 | — | IC50 | = | 51973.97 | nM | 4.28 |
| CHEMBL258844 | — | IC50 | = | 57143.69 | nM | 4.24 |