Assay Detail
Functional
CHEMBL2363240
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human GCT cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | GCT |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.45 | 8.74 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.74 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.32 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.30 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.28 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.18 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.86 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.63 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.38 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.29 |
| CHEMBL217354 | — | — | 1 | 6.72 |
| CHEMBL585951 | — | — | 1 | 6.69 |
| CHEMBL412142 | LADUVIGLUSIB | 1.0 | 1 | 6.51 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.49 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 6.39 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.28 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.19 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.19 |
| CHEMBL1190711 | — | — | 1 | 6.10 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.07 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.07 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.94 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.87 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 5.70 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 5.66 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 5.64 |
| CHEMBL573107 | — | — | 1 | 5.64 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 5.59 |
| CHEMBL2363137 | — | — | 1 | 5.53 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 5.49 |
| CHEMBL191384 | — | — | 1 | 5.44 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.797 | nM | 8.74 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 4.728 | nM | 8.32 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 5.023 | nM | 8.30 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 5.303 | nM | 8.28 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 6.612 | nM | 8.18 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 13.68 | nM | 7.86 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 23.39 | nM | 7.63 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 41.61 | nM | 7.38 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 50.77 | nM | 7.29 |
| CHEMBL217354 | — | IC50 | = | 191.13 | nM | 6.72 |
| CHEMBL585951 | — | IC50 | = | 203.9 | nM | 6.69 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 306.72 | nM | 6.51 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 326.93 | nM | 6.49 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 405.1 | nM | 6.39 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 528.97 | nM | 6.28 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 641.53 | nM | 6.19 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 649.35 | nM | 6.19 |
| CHEMBL1190711 | — | IC50 | = | 798.87 | nM | 6.10 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 861.48 | nM | 6.07 |
| CHEMBL803 | CYTARABINE | IC50 | = | 855.68 | nM | 6.07 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1151.53 | nM | 5.94 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1343.45 | nM | 5.87 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 2009.16 | nM | 5.70 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 2177.7 | nM | 5.66 |
| CHEMBL573107 | — | IC50 | = | 2313.58 | nM | 5.64 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 2303.04 | nM | 5.64 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 2586.94 | nM | 5.59 |
| CHEMBL2363137 | — | IC50 | = | 2929.27 | nM | 5.53 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 3265.76 | nM | 5.49 |
| CHEMBL191384 | — | IC50 | = | 3597.3 | nM | 5.44 |
| CHEMBL202721 | — | IC50 | = | 3769.8 | nM | 5.42 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 4104.42 | nM | 5.39 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 4604.7 | nM | 5.34 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 4990.65 | nM | 5.30 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 5246.26 | nM | 5.28 |
| CHEMBL521686 | OLAPARIB | IC50 | = | 5568.56 | nM | 5.25 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 5759.29 | nM | 5.24 |
| CHEMBL393929 | — | IC50 | = | 5851.21 | nM | 5.23 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 5997.11 | nM | 5.22 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 6122.44 | nM | 5.21 |
| CHEMBL939 | GEFITINIB | IC50 | = | 6533.87 | nM | 5.18 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 6736.81 | nM | 5.17 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 6938.0 | nM | 5.16 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 6960.0 | nM | 5.16 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 7569.06 | nM | 5.12 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 7821.72 | nM | 5.11 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 8753.14 | nM | 5.06 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 9098.31 | nM | 5.04 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 10112.19 | nM | 5.00 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 11822.75 | nM | 4.93 |