Assay Detail
Functional
CHEMBL2363247
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SANGER: Inhibition of human GR-ST cell growth in a cell viability assay.
130
Total Activities
129
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | GR-ST |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 130 | 5.73 | 10.23 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 10.23 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 9.19 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.15 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 9.07 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.41 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.12 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.08 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.98 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.58 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 7.50 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.48 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.44 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.28 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.25 |
| CHEMBL514499 | GW843682X | — | 1 | 7.08 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.99 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 6.99 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 6.95 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.92 |
| CHEMBL300389 | — | — | 1 | 6.76 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.75 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 6.67 |
| CHEMBL512504 | — | — | 1 | 6.66 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.59 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.42 |
| CHEMBL379300 | A-443654 | — | 1 | 6.35 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.31 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.28 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.20 |
| CHEMBL585951 | — | — | 1 | 6.19 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.05953 | nM | 10.23 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 0.648 | nM | 9.19 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.701 | nM | 9.15 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 0.8457 | nM | 9.07 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 3.907 | nM | 8.41 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 7.631 | nM | 8.12 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 8.272 | nM | 8.08 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 10.5 | nM | 7.98 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 26.55 | nM | 7.58 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 31.85 | nM | 7.50 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 33.35 | nM | 7.48 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 36.28 | nM | 7.44 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 52.87 | nM | 7.28 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 56.21 | nM | 7.25 |
| CHEMBL514499 | GW843682X | IC50 | = | 83.98 | nM | 7.08 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 102.18 | nM | 6.99 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 102.1 | nM | 6.99 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 113.34 | nM | 6.95 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 121.34 | nM | 6.92 |
| CHEMBL300389 | — | IC50 | = | 174.08 | nM | 6.76 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 178.27 | nM | 6.75 |
| CHEMBL513909 | BI-2536 | IC50 | = | 214.88 | nM | 6.67 |
| CHEMBL512504 | — | IC50 | = | 217.64 | nM | 6.66 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 255.42 | nM | 6.59 |
| CHEMBL803 | CYTARABINE | IC50 | = | 384.72 | nM | 6.42 |
| CHEMBL379300 | A-443654 | IC50 | = | 448.37 | nM | 6.35 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 493.74 | nM | 6.31 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 530.15 | nM | 6.28 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 628.3 | nM | 6.20 |
| CHEMBL585951 | — | IC50 | = | 647.47 | nM | 6.19 |
| CHEMBL36 | PYRIMETHAMINE | IC50 | = | 708.82 | nM | 6.15 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 872.37 | nM | 6.06 |
| CHEMBL379975 | — | IC50 | = | 975.21 | nM | 6.01 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 1094.29 | nM | 5.96 |
| CHEMBL509032 | TAE-684 | IC50 | = | 1387.57 | nM | 5.86 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1568.2 | nM | 5.80 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 2874.57 | nM | 5.54 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 2965.85 | nM | 5.53 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 3046.11 | nM | 5.52 |
| CHEMBL401930 | — | IC50 | = | 3271.56 | nM | 5.49 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 3221.39 | nM | 5.49 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 3457.32 | nM | 5.46 |
| CHEMBL64925 | MG-132 | IC50 | = | 3592.66 | nM | 5.45 |
| CHEMBL1190711 | — | IC50 | = | 3698.6 | nM | 5.43 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 4176.35 | nM | 5.38 |
| CHEMBL939 | GEFITINIB | IC50 | = | 4431.8 | nM | 5.35 |
| CHEMBL577784 | BX-795 | IC50 | = | 4978.5 | nM | 5.30 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 5383.22 | nM | 5.27 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 5522.01 | nM | 5.26 |
| CHEMBL259181 | — | IC50 | = | 5505.01 | nM | 5.26 |