Assay Detail
Functional
CHEMBL2363252
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SANGER: Inhibition of human HAL-01 cell growth in a cell viability assay.
130
Total Activities
129
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HAL-01 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 130 | 5.68 | 9.34 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 9.34 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.93 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.59 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 8.53 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.30 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.09 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.80 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.65 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.25 |
| CHEMBL300389 | — | — | 1 | 7.18 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.12 |
| CHEMBL514499 | GW843682X | — | 1 | 7.09 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.89 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.71 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.69 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.68 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.68 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 6.63 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.52 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.51 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.50 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.48 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 6.41 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.34 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.33 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.22 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 6.21 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 6.18 |
| CHEMBL585951 | — | — | 1 | 6.15 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 6.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 0.4527 | nM | 9.34 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 1.182 | nM | 8.93 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 2.551 | nM | 8.59 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 2.968 | nM | 8.53 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 5.017 | nM | 8.30 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 8.195 | nM | 8.09 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 15.73 | nM | 7.80 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 22.27 | nM | 7.65 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 55.83 | nM | 7.25 |
| CHEMBL300389 | — | IC50 | = | 66.04 | nM | 7.18 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 76.58 | nM | 7.12 |
| CHEMBL514499 | GW843682X | IC50 | = | 80.77 | nM | 7.09 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 128.09 | nM | 6.89 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 195.73 | nM | 6.71 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 202.97 | nM | 6.69 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 206.73 | nM | 6.68 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 209.7 | nM | 6.68 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 233.41 | nM | 6.63 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 300.96 | nM | 6.52 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 306.46 | nM | 6.51 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 313.44 | nM | 6.50 |
| CHEMBL803 | CYTARABINE | IC50 | = | 327.86 | nM | 6.48 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 389.26 | nM | 6.41 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 454.12 | nM | 6.34 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 469.09 | nM | 6.33 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 605.67 | nM | 6.22 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 621.3 | nM | 6.21 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 662.2 | nM | 6.18 |
| CHEMBL585951 | — | IC50 | = | 703.97 | nM | 6.15 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 725.49 | nM | 6.14 |
| CHEMBL939 | GEFITINIB | IC50 | = | 734.71 | nM | 6.13 |
| CHEMBL591429 | PAC-1 | IC50 | = | 788.3 | nM | 6.10 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 968.04 | nM | 6.01 |
| CHEMBL513909 | BI-2536 | IC50 | = | 998.72 | nM | 6.00 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 993.79 | nM | 6.00 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 1088.1 | nM | 5.96 |
| CHEMBL401930 | — | IC50 | = | 1123.1 | nM | 5.95 |
| CHEMBL509032 | TAE-684 | IC50 | = | 1152.83 | nM | 5.94 |
| CHEMBL379975 | — | IC50 | = | 1160.02 | nM | 5.94 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1169.43 | nM | 5.93 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 1167.09 | nM | 5.93 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1301.75 | nM | 5.88 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 1695.7 | nM | 5.77 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 1711.47 | nM | 5.77 |
| CHEMBL535 | SUNITINIB | IC50 | = | 2059.46 | nM | 5.69 |
| CHEMBL1673039 | — | IC50 | = | 2115.17 | nM | 5.67 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 2420.77 | nM | 5.62 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 2742.49 | nM | 5.56 |
| CHEMBL477989 | SB590885 | IC50 | = | 2925.79 | nM | 5.53 |
| CHEMBL197603 | — | IC50 | = | 3082.64 | nM | 5.51 |