Assay Detail
Functional
CHEMBL2363439
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SANGER: Inhibition of human MONO-MAC-6 cell growth in a cell viability assay.
78
Total Activities
77
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MONO-MAC-6 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 78 | 5.94 | 8.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.51 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.42 |
| CHEMBL1336 | SORAFENIB | 4.0 | 1 | 8.38 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 8.08 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.76 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.69 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.61 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.52 |
| CHEMBL535 | SUNITINIB | 4.0 | 1 | 7.47 |
| CHEMBL514499 | GW843682X | — | 1 | 7.46 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.41 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.14 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.14 |
| CHEMBL379300 | A-443654 | — | 1 | 7.11 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.10 |
| CHEMBL572878 | TOZASERTIB | 2.0 | 1 | 7.10 |
| CHEMBL300389 | — | — | 1 | 7.07 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.98 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.95 |
| CHEMBL512504 | — | — | 1 | 6.94 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.81 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.61 |
| CHEMBL509032 | TAE-684 | — | 1 | 6.48 |
| CHEMBL27759 | ENTINOSTAT | 3.0 | 1 | 6.41 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.36 |
| CHEMBL64925 | MG-132 | — | 2 | 6.27 |
| CHEMBL585951 | — | — | 1 | 6.26 |
| CHEMBL401930 | — | — | 1 | 6.22 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 6.12 |
| CHEMBL1190711 | — | — | 1 | 6.02 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 3.104 | nM | 8.51 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 3.801 | nM | 8.42 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 4.181 | nM | 8.38 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 8.372 | nM | 8.08 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 17.36 | nM | 7.76 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 20.61 | nM | 7.69 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 24.84 | nM | 7.61 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 30.23 | nM | 7.52 |
| CHEMBL535 | SUNITINIB | IC50 | = | 33.8 | nM | 7.47 |
| CHEMBL514499 | GW843682X | IC50 | = | 34.64 | nM | 7.46 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 38.93 | nM | 7.41 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 72.12 | nM | 7.14 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 72.35 | nM | 7.14 |
| CHEMBL379300 | A-443654 | IC50 | = | 77.23 | nM | 7.11 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 78.79 | nM | 7.10 |
| CHEMBL513909 | BI-2536 | IC50 | = | 79.86 | nM | 7.10 |
| CHEMBL300389 | — | IC50 | = | 85.87 | nM | 7.07 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 104.95 | nM | 6.98 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 111.36 | nM | 6.95 |
| CHEMBL512504 | — | IC50 | = | 113.72 | nM | 6.94 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 154.36 | nM | 6.81 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 244.77 | nM | 6.61 |
| CHEMBL509032 | TAE-684 | IC50 | = | 332.91 | nM | 6.48 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 387.76 | nM | 6.41 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 438.49 | nM | 6.36 |
| CHEMBL64925 | MG-132 | IC50 | = | 536.11 | nM | 6.27 |
| CHEMBL585951 | — | IC50 | = | 543.72 | nM | 6.26 |
| CHEMBL401930 | — | IC50 | = | 607.94 | nM | 6.22 |
| CHEMBL64925 | MG-132 | IC50 | = | 718.2 | nM | 6.14 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 756.93 | nM | 6.12 |
| CHEMBL1190711 | — | IC50 | = | 963.1 | nM | 6.02 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 1153.51 | nM | 5.94 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 1180.97 | nM | 5.93 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 2132.31 | nM | 5.67 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 2412.48 | nM | 5.62 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 3348.94 | nM | 5.47 |
| CHEMBL515416 | — | IC50 | = | 3926.1 | nM | 5.41 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 4593.84 | nM | 5.34 |
| CHEMBL258844 | — | IC50 | = | 4747.75 | nM | 5.32 |
| CHEMBL2363137 | — | IC50 | = | 6182.57 | nM | 5.21 |
| CHEMBL209148 | — | IC50 | = | 6667.79 | nM | 5.18 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 8270.66 | nM | 5.08 |
| CHEMBL180127 | SALUBRINAL | IC50 | = | 10548.25 | nM | 4.98 |
| CHEMBL259181 | — | IC50 | = | 10404.17 | nM | 4.98 |
| CHEMBL1643959 | — | IC50 | = | 12099.75 | nM | 4.92 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 12130.88 | nM | 4.92 |
| CHEMBL591429 | PAC-1 | IC50 | = | 11902.29 | nM | 4.92 |
| CHEMBL191384 | — | IC50 | = | 12617.23 | nM | 4.90 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 14150.19 | nM | 4.85 |
| CHEMBL36 | PYRIMETHAMINE | IC50 | = | 16286.2 | nM | 4.79 |