Assay Detail
Functional
CHEMBL2363553
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SANGER: Inhibition of human NCI-SNU-1 cell growth in a cell viability assay.
130
Total Activities
129
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SNU1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 130 | 5.73 | 10.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 10.80 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.96 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.79 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.71 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 8.68 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 8.32 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.31 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 8.12 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 7.88 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.87 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.66 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.49 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.20 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.18 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.10 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 7.01 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 7.01 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.92 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.81 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.74 |
| CHEMBL300389 | — | — | 1 | 6.58 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.57 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.55 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 6.53 |
| CHEMBL512504 | — | — | 1 | 6.51 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.49 |
| CHEMBL379300 | A-443654 | — | 1 | 6.40 |
| CHEMBL2144069 | — | — | 1 | 6.35 |
| CHEMBL585951 | — | — | 1 | 6.34 |
| CHEMBL188678 | — | — | 1 | 6.21 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.01596 | nM | 10.80 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 1.088 | nM | 8.96 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 1.622 | nM | 8.79 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.969 | nM | 8.71 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 2.068 | nM | 8.68 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 4.806 | nM | 8.32 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 4.862 | nM | 8.31 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 7.515 | nM | 8.12 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 13.19 | nM | 7.88 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 13.59 | nM | 7.87 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 21.95 | nM | 7.66 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 32.75 | nM | 7.49 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 62.74 | nM | 7.20 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 65.86 | nM | 7.18 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 78.88 | nM | 7.10 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 96.73 | nM | 7.01 |
| CHEMBL803 | CYTARABINE | IC50 | = | 96.77 | nM | 7.01 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 121.48 | nM | 6.92 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 156.24 | nM | 6.81 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 183.41 | nM | 6.74 |
| CHEMBL300389 | — | IC50 | = | 260.56 | nM | 6.58 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 270.59 | nM | 6.57 |
| CHEMBL939 | GEFITINIB | IC50 | = | 283.32 | nM | 6.55 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 294.22 | nM | 6.53 |
| CHEMBL512504 | — | IC50 | = | 311.06 | nM | 6.51 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 323.31 | nM | 6.49 |
| CHEMBL379300 | A-443654 | IC50 | = | 400.14 | nM | 6.40 |
| CHEMBL2144069 | — | IC50 | = | 447.86 | nM | 6.35 |
| CHEMBL585951 | — | IC50 | = | 458.16 | nM | 6.34 |
| CHEMBL188678 | — | IC50 | = | 609.94 | nM | 6.21 |
| CHEMBL393929 | — | IC50 | = | 730.95 | nM | 6.14 |
| CHEMBL105442 | CI-1040 | IC50 | = | 754.33 | nM | 6.12 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 772.78 | nM | 6.11 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 828.82 | nM | 6.08 |
| CHEMBL379975 | — | IC50 | = | 897.88 | nM | 6.05 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 1023.31 | nM | 5.99 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1163.54 | nM | 5.93 |
| CHEMBL3349342 | — | IC50 | = | 1241.37 | nM | 5.91 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 1330.4 | nM | 5.88 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 1365.55 | nM | 5.87 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1602.2 | nM | 5.79 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1753.27 | nM | 5.76 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 1772.43 | nM | 5.75 |
| CHEMBL1190711 | — | IC50 | = | 1990.98 | nM | 5.70 |
| CHEMBL189584 | PD-173074 | IC50 | = | 2183.94 | nM | 5.66 |
| CHEMBL509032 | TAE-684 | IC50 | = | 2332.56 | nM | 5.63 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 2316.2 | nM | 5.63 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 2703.25 | nM | 5.57 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 2690.28 | nM | 5.57 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 2840.84 | nM | 5.55 |